SCHEMBL9750127

SCHEMBL9750127

C=C1N(C)c2c(Oc3ccccc3)cccc2C1(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.34
ALDH1A1 P00352 3/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
HPGD P15428 2/20 0.33
RIPK1 Q13546 1/20 0.33
LMNA P02545 2/20 0.33
KMT2A Q03164 2/20 0.33
DPP4 P27487 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN3A Q9NY46 1/20 0.32
LTA4H P09960 1/20 0.31
TSHR P16473 1/20 0.31
TSPO P30536 1/20 0.31
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750033 0.89 ALDH1A1 (0.38) ALDH1A1SLC6A2SLC6A4HPGDLMNA
SCHEMBL9750451 0.86 ALDH1A1 (0.44) ALDH1A1LMNAKMT2AGAAHTT
SCHEMBL9750256 0.81 ALDH1A1 (0.35) ALDH1A1SLC6A2SLC6A4HPGDLMNA
SCHEMBL9750259 0.79 MAPT (0.46) BRD4ALDH1A1HPGDKMT2AGAA
SCHEMBL9750191 0.78 PDK2 (0.39) ALDH1A1HPGDLMNAKMT2AGAA
SCHEMBL4603103 0.73 MEN1 (0.37) ALDH1A1LMNAKMT2AGAAHTT
SCHEMBL11019576 0.72 MAPT (0.46) ALDH1A1HPGDLMNAKMT2AGAA
SCHEMBL9750080 0.71 ALDH1A1 (0.39) ALDH1A1HPGDLMNAKMT2AMAPK1
SCHEMBL9750447 0.71 PGR (0.33) ALDH1A1LMNAMAPK1L3MBTL1MAPT
SCHEMBL8942200 0.71 GRIA2 (0.42) LMNAMAPK1HTTLTA4HTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172892-A Heteromonocyclic and heterobicyclic derivatives of unsaturated 7-acylamido-3-cephem-4-carboxylic acid CARLO ERBA S.P.A. (IT) 1979-10-30 US claimed
US-5120858-A Condensation of 2-methyleneindoline and formic acid in acetic anhydride MILES INC. (US) 1992-06-09 US disclosed
EP-0058863-B1 PROCESS FOR THE PREPARATION OF TRIMETHINE DYESTUFFS BAYER AG (DE) 1985-01-23 EP disclosed
EP-0113920-A2 Process for the manufacture of stable solutions of cationic methine dyes, and their use in spin dyeing BAYER AG (DE) 1984-07-25 EP disclosed
US-4419511-A Process for the preparation of trimethine dyestuffs BAYER AKTIENGESELLSCHAFT (US) 1983-12-06 US disclosed
US-4388314-A BACTERICIDES FARMITALIA CARLO ERBA S.P.A. (IT) 1983-06-14 US disclosed
EP-0058863-A1 Process for the preparation of trimethine dyestuffs BAYER AG (DE) 1982-09-01 EP disclosed
US-4172892-A Heteromonocyclic and heterobicyclic derivatives of unsaturated 7-acylamido-3-cephem-4-carboxylic acid CARLO ERBA S.P.A. (IT) 1979-10-30 US disclosed