SCHEMBL9750187

SCHEMBL9750187

C=C1N(C)c2c(CC)cccc2C1(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.42
NPEPPS P55786 2/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
GABRA1 P14867 3/20 0.34
GABRB2 P47870 3/20 0.34
LMNA P02545 2/20 0.34
HTT P42858 2/20 0.34
MAPT P10636 2/20 0.34
MPI P34949 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP2D6 P10635 1/20 0.33
ANPEP P15144 2/20 0.32
DPP4 P27487 2/20 0.32
TSHR P16473 2/20 0.31
MEN1 O00255 1/20 0.31
THRB P10828 1/20 0.31
RECQL P46063 1/20 0.31
KMT2A Q03164 1/20 0.31
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4603103 0.77 MEN1 (0.37) LMNAHTTMAPTMPITDP1
SCHEMBL9750191 0.76 PDK2 (0.39) PDK2LMNAMAPTTDP1MEN1
SCHEMBL10938890 0.73 GABRA1 (0.34) GABRA1GABRB2LMNAMPITDP1
SCHEMBL9750256 0.73 ALDH1A1 (0.35) PDK2LMNAHTTMAPTMEN1
SCHEMBL11019576 0.71 MAPT (0.46) LMNAHTTMAPTTDP1TSHR
SCHEMBL9750259 0.69 MAPT (0.46) MAPTTDP1MEN1KMT2AHTR1A
SCHEMBL9750127 0.69 BRD4 (0.34) LMNAHTTMAPTTDP1DPP4
Alcohol SCHEMBL27668500 0.68 MAPT (0.45) CRHBPCRHR2LMNAHTTMAPT
SCHEMBL9750080 0.67 ALDH1A1 (0.39) LMNAHTTMAPTTDP1CYP2D6
SCHEMBL918366 0.67 HTT (0.51) CRHBPCRHR2LMNAHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120858-A Condensation of 2-methyleneindoline and formic acid in acetic anhydride MILES INC. (US) 1992-06-09 US disclosed
EP-0058863-B1 PROCESS FOR THE PREPARATION OF TRIMETHINE DYESTUFFS BAYER AG (DE) 1985-01-23 EP disclosed
US-4419511-A Process for the preparation of trimethine dyestuffs BAYER AKTIENGESELLSCHAFT (US) 1983-12-06 US disclosed
US-4201707-A Methine dyestuffs containing a phenyl azo group BAYER AKTIENGESELLSCHAFT (DE) 1980-05-06 US disclosed
US-4143228-A RED SHADES BAYER AKTIENGESELLSCHAFT (DE) 1979-03-06 US disclosed
US-4138570-A METHINE DYE BAYER AKTIENGESELLSCHAFT (DE) 1979-02-06 US disclosed