SCHEMBL9518155

SCHEMBL9518155

CC(C)c1c(/C=C/C#N)c(-c2ccc(F)cc2)cn1C(C)C

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 7/20 0.53
TGFBR1 P36897 2/20 0.34
NR3C1 P04150 2/20 0.32
PGR P06401 2/20 0.32
NR3C2 P08235 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
AR P10275 1/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
TGFBR2 P37173 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9518437 0.82 HMGCR (0.56) HMGCRMAPK13MAPK12MAPK11MAPK14
SCHEMBL9750945 0.82 HMGCR (0.56) HMGCRMAPK13MAPK12MAPK11MAPK14
SCHEMBL9751046 0.81 HMGCR (0.55) HMGCRALDH1A1MAPK13MAPK12MAPK11
SCHEMBL9518598 0.80 HMGCR (0.56) HMGCRTGFBR1MAPK13MAPK12MAPK11
SCHEMBL9024469 0.75 PKM (0.38) HMGCRKDM4EALDH1A1SMN1; SMN2
SCHEMBL9750874 0.73 HMGCR (0.41) HMGCRTGFBR1KDM4EALDH1A1GAA
SCHEMBL9024739 0.72 NR4A2 (0.34) NR3C1PGRNR3C2KDM4EALDH1A1
SCHEMBL9518177 0.71 HMGCR (0.47) HMGCR
SCHEMBL9764350 0.71 KDM4E (0.43) HMGCRKDM4EALDH1A1
SCHEMBL9518302 0.70 HMGCR (0.66) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0300249-B1 7-[1H-pyrrol-3-yl]-substituted 3,5-dihydroxy-heptane acids, their corresponding delta-lactones and salts, processes for their manufacture, their use as medicines, pharmaceutical preparations and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1993-02-03 EP disclosed
US-5055484-A Anticholesterol and antilipemic agent HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-08 US disclosed
EP-0300249-A1 7-[1H-pyrrol-3-yl]-substituted 3,5-dihydroxy-heptane acids, their corresponding delta-lactones and salts, processes for their manufacture, their use as medicines, pharmaceutical preparations and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1989-01-25 EP disclosed