SCHEMBL9753315

SCHEMBL9753315

CC(=O)OCc1c(-c2ccc(F)cc2)nn2cccc2c1C(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.39
EGFR P00533 2/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
RAF1 P04049 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
GSK3B P49841 1/20 0.39
PTGS2 P35354 2/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
MIF P14174 2/20 0.34
KCNK3 O14649 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753170 0.83 MAPK14 (0.44) MAPK14EGFRADORA2AADORA1RAF1
SCHEMBL9752865 0.79 ALDH1A1 (0.49) MAPK14EGFRADORA2AADORA1RAF1
SCHEMBL9752965 0.78 MAPK14 (0.43) MAPK14EGFRADORA2AADORA1RAF1
SCHEMBL9752947 0.75 HMGCR (0.49) HMGCR
SCHEMBL9753321 0.74 MAPK14 (0.44) MAPK14EGFRADORA2AADORA1RAF1
SCHEMBL9752919 0.72 SMN1; SMN2 (0.43) EGFRADORA2AADORA1MEN1KMT2A
SCHEMBL9753346 0.71 GCGR (0.39) MAPK14EGFRADORA2AADORA1RAF1
SCHEMBL9753160 0.70 MAPK14 (0.41) MAPK14EGFRADORA2AADORA1RAF1
SCHEMBL9753157 0.70 MAPK14 (0.41) MAPK14EGFRADORA2AADORA1RAF1
SCHEMBL9752979 0.70 KDM4E (0.51) EGFRADORA3MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed
CN-1056690-A PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO (JP) 1991-12-04 CN disclosed