SCHEMBL9753346

SCHEMBL9753346

CC(C)c1c(CO)c(-c2ccc(F)c(F)c2)nn2cccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 4/20 0.39
TGFBR1 P36897 2/20 0.33
MAPK14 Q16539 2/20 0.32
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
EGFR P00533 1/20 0.32
RAF1 P04049 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2B P29275 1/20 0.32
GSK3B P49841 1/20 0.32
GRIN2B Q13224 2/20 0.32
MIF P14174 2/20 0.32
TRPV3 Q8NET8 1/20 0.32
RAD51 Q06609 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
GRIN1 Q05586 1/20 0.31
GABRA5 P31644 1/20 0.31
MEN1 O00255 1/20 0.31
PDE5A O76074 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753002 0.90 TGFBR1 (0.36) TGFBR1MAPK14ADORA2AADORA1EGFR
SCHEMBL9753170 0.87 MAPK14 (0.44) GCGRMAPK14ADORA2AADORA1EGFR
SCHEMBL9752919 0.83 SMN1; SMN2 (0.43) GCGRADORA2AADORA1EGFRMIF
SCHEMBL9753098 0.81 GCGR (0.40) GCGRTGFBR1MAPK14ADORA2AADORA1
SCHEMBL9753354 0.79 PTGS2 (0.34) TGFBR1MAPK14ADORA2AADORA1EGFR
SCHEMBL9753377 0.78 EGFR (0.44) ADORA2AADORA1EGFRMIFMEN1
SCHEMBL9753419 0.76 GRM2 (0.36) GCGRMAPK14
SCHEMBL9753721 0.76 PTGS2 (0.32) MAPK14ADORA2AADORA1EGFRRAF1
SCHEMBL9753724 0.76 PTGS2 (0.32) MAPK14ADORA2AADORA1EGFRRAF1
SCHEMBL9753097 0.71 HMGCR (0.45) ADORA3ALDH1A1CYP3A4CYP2C9PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed