SCHEMBL9754431

SCHEMBL9754431

O=c1[nH]c(-c2cc3ccccc3o2)ccc1-c1nnn[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.45
NPC1 O15118 3/20 0.45
SIRT1 Q96EB6 1/20 0.43
PDE10A Q9Y233 1/20 0.40
PTPRC P08575 1/20 0.40
PTPN1 P18031 1/20 0.40
ADRA2A P08913 2/20 0.39
GPR35 Q9HC97 1/20 0.38
KDM5A P29375 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.37
MAOB P27338 4/20 0.36
MAOA P21397 2/20 0.36
METAP2 P50579 1/20 0.36
NPY5R Q15761 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31652715 0.79 ADRA2A (0.54) RAB9ANPC1PTPRCPTPN1ADRA2A
SCHEMBL11018706 0.77 GPR35 (0.58) RAB9ANPC1GPR35KDM4EALDH1A1
SCHEMBL9754365 0.77 ALDH1A1 (0.36) RAB9ANPC1SIRT1KDM4EALDH1A1
SCHEMBL9251638 0.77 PTGER3 (0.46)
SCHEMBL9535284 0.75 KDM4E (0.41) PDE10AKDM4E
SCHEMBL9754436 0.74 ALDH1A1 (0.33) RAB9ANPC1KDM4EALDH1A1HPGD
SCHEMBL9754463 0.74 PTGER3 (0.39)
SCHEMBL9754374 0.73 NPC1 (0.40) RAB9ANPC1KDM4EALDH1A1MAPT
SCHEMBL12496454 0.70 NPC1 (0.40) RAB9ANPC1ADRA2AGPR35KDM4E
SCHEMBL7499608 0.70 KDR (0.60) RAB9ANPC1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO claimed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed