SCHEMBL9764516

SCHEMBL9764516

Nc1c(Cl)cc(C(O)CN(CCCCCCOCCc2ccc(N3CCOCC3)cc2)Cc2ccccc2)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.37
ADRB2 P07550 1/20 0.35
AOC3 Q16853 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
MAPT P10636 2/20 0.33
SLC2A1 P11166 1/20 0.33
NAMPT P43490 1/20 0.33
SIGMAR1 Q99720 2/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
GAA P10253 1/20 0.32
NAPEPLD Q6IQ20 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764456 0.88 ADRB2 (0.41) ADRB2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL9764429 0.88 ADRB2 (0.41) ADRB2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL9764329 0.85 ADRB2 (0.39) ADRB2SLC6A2SLC6A4SLC6A3SLC2A1
SCHEMBL9764389 0.85 ADRB2 (0.39) ADRB2MAPTSLC2A1
SCHEMBL9764371 0.85 ADRB2 (0.41) ADRB2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL9764694 0.83 NR1H3 (0.45) ADRB2
SCHEMBL9764242 0.81 MC4R (0.39) ADRB2
SCHEMBL9321535 0.80 MAOB (0.37) ADRB2CYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL9764301 0.80 NR1H3 (0.45) ADRB2
SCHEMBL10423748 0.80 ADRB2 (0.41) ADRB2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed
EP-0181709-A1 Dichloroaniline Derivatives GLAXO GROUP LIMITED (GB) 1986-05-21 EP disclosed