SCHEMBL9764538

SCHEMBL9764538

CCOC(=O)c1ccc(C#CCOCCCCCCN(Cc2ccccc2)CC(O)c2cc(Cl)c(N)c(Cl)c2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.35
TP53 P04637 1/20 0.35
BCHE P06276 3/20 0.35
ACHE P22303 3/20 0.35
MMP2 P08253 2/20 0.35
MMP12 P39900 2/20 0.35
KDM4E B2RXH2 3/20 0.33
POLB P06746 1/20 0.33
MAOB P27338 3/20 0.33
MAPT P10636 3/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764279 0.90 NR1H3 (0.35) BCHEACHEMMP2MMP12KDM4E
SCHEMBL10466598 0.88 MMP13 (0.34) BCHEACHEKDM4EMAOBMEN1
SCHEMBL10469272 0.88 HPGD (0.33) HPGDTP53BCHEACHEKDM4E
SCHEMBL9764533 0.85 HPGD (0.35) HPGDTP53BCHEACHEMMP2
SCHEMBL9764569 0.84 SNCA (0.38) HPGDALDH1A1KMT2A
SCHEMBL10468372 0.84 NR1H3 (0.33) BCHEACHEKDM4EMAPTALDH1A1
SCHEMBL9764548 0.84 KCNH2 (0.33) BCHEACHEKDM4ENR1H3
SCHEMBL9764422 0.83 LTA4H (0.37) KDM4EPOLBMAPTALDH1A1HTT
SCHEMBL10466615 0.83 NR1H3 (0.34) BCHEACHEKDM4EMAOBMEN1
SCHEMBL9319139 0.82 MAOB (0.38) MAOBALDH1A1NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed
EP-0181709-A1 Dichloroaniline Derivatives GLAXO GROUP LIMITED (GB) 1986-05-21 EP disclosed