SCHEMBL9768831

SCHEMBL9768831

CN1c2ccccc2N(C(=O)CN2CCCC2)c2ccccc2S1(=O)=O

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
USP2 O75604 2/20 0.56
ALOX15 P16050 1/20 0.56
TP53 P04637 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HTT P42858 1/20 0.42
GAA P10253 1/20 0.42
POLB P06746 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PKM P14618 1/20 0.42
NR1I3 Q14994 2/20 0.42
RAD52 P43351 1/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768740 0.92 CYP2D6 (0.53) ALDH1A1USP2ALOX15TP53CYP3A4
Hydrochloric Acid SCHEMBL9768751 0.88 ALDH1A1 (0.44) ALDH1A1USP2ALOX15TP53CYP3A4
SCHEMBL9768745 0.88 TP53 (0.62) ALDH1A1USP2ALOX15TP53CYP3A4
SCHEMBL9768785 0.81 NPC1 (0.53) ALDH1A1TP53HTT
SCHEMBL9768706 0.78 MAPT (0.44) ALDH1A1TP53KMT2AHTTKDM4E
SCHEMBL9768762 0.78 NPC1 (0.40) ALDH1A1TP53MEN1KMT2AHTT
SCHEMBL9768832 0.78 MTNR1A (0.40) TP53CYP3A4MEN1KMT2AHTT
SCHEMBL9768739 0.78 GRM7 (0.38) ALDH1A1TP53CYP3A4CYP2D6MEN1
SCHEMBL9768744 0.76 NR1I3 (0.44) ALDH1A1TP53CYP2D6GAAPOLB
SCHEMBL9768823 0.76 KDM4E (0.46) ALDH1A1TP53MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011833-A Antidepressant A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE (IT) 1991-04-30 US disclosed
EP-0354885-A1 Novel derivatives of 6,11-dihydro-dibenzo[c,f][1,2,5]-thiadiazepine 5,5-dioxide, salts thereof and appropriate processes for the preparation thereof A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1990-02-14 EP disclosed