SCHEMBL9768744

SCHEMBL9768744

CCN(CC)CC(=O)N1c2ccccc2N(C)S(=O)(=O)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1I3 Q14994 10/20 0.44
GAA P10253 1/20 0.42
KDM4E B2RXH2 2/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
POLB P06746 1/20 0.40
CACNA1C Q13936 1/20 0.38
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768706 0.86 MAPT (0.44) NR1I3KDM4EMAPTSMN1; SMN2ALDH1A1
SCHEMBL9768785 0.81 NPC1 (0.53) ALDH1A1TP53
SCHEMBL9768823 0.79 KDM4E (0.46) NR1I3KDM4EMAPTPOLBALDH1A1
SCHEMBL9768762 0.78 NPC1 (0.40) MAPTALDH1A1TP53
SCHEMBL9768832 0.78 MTNR1A (0.40) GAAMAPTPOLBTP53
Hydrochloric Acid SCHEMBL9768695 0.78 KDM4E (0.47) NR1I3KDM4EMAPTSMN1; SMN2POLB
SCHEMBL9768826 0.77 MAPT (0.41) NR1I3GAAKDM4ECYP2D6MAPT
SCHEMBL9768831 0.76 ALDH1A1 (0.56) NR1I3GAAKDM4ECYP2D6MAPT
SCHEMBL9768740 0.76 CYP2D6 (0.53) NR1I3KDM4ECYP2D6MAPTALDH1A1
SCHEMBL9768774 0.76 ALDH1A1 (0.43) NR1I3KDM4ECYP2D6MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011833-A Antidepressant A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE (IT) 1991-04-30 US claimed
US-5011833-A Antidepressant A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE (IT) 1991-04-30 US disclosed
EP-0354885-A1 Novel derivatives of 6,11-dihydro-dibenzo[c,f][1,2,5]-thiadiazepine 5,5-dioxide, salts thereof and appropriate processes for the preparation thereof A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1990-02-14 EP disclosed