SCHEMBL9769828

SCHEMBL9769828

CCOC(=O)C(=C(c1ccc(F)cc1)c1ccc(F)cc1)n1nnnc1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 3/20 0.42
MGLL Q99685 1/20 0.41
TP53 P04637 1/20 0.40
HSD11B1 P28845 2/20 0.39
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CYP19A1 P11511 1/20 0.38
NR3C2 P08235 1/20 0.38
TSHR P16473 1/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9769861 0.85 HMGCR (0.45) ELANEALDH1A1HPGDNPSR1TP53
SCHEMBL9769894 0.75 ALDH1A1 (0.43) ALDH1A1HPGDMGLLHSD11B1PKM
SCHEMBL9769831 0.74 ALDH1A1 (0.42) ALDH1A1HPGDMGLLHSD11B1PKM
SCHEMBL9769919 0.73 HMGCR (0.61)
SCHEMBL9769922 0.73 HMGCR (0.61)
SCHEMBL9769858 0.73 HMGCR (0.51) ELANEALDH1A1HPGDNPSR1SMN1; SMN2
SCHEMBL9769851 0.73 HMGCR (0.51) ELANEALDH1A1HPGDNPSR1SMN1; SMN2
SCHEMBL9769860 0.73 HMGCR (0.42) ELANEALDH1A1HPGDNPSR1PKM
SCHEMBL12781922 0.71 MGLL (0.51) ELANEALDH1A1HPGDMGLLHSD11B1
SCHEMBL9769841 0.70 HMGCR (0.41) ALDH1A1HPGDMGLLHSD11B1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070206-A INHIBITORS OF 3-HYDROXY-3-METHYLGLUTARYL COENZYME A REDUCTASE; ANTICHOLESTEROL, ANTILIPEMIC BRISTOL-MYERS COMPANY (US) 1991-12-03 US disclosed
US-5010205-A Antihypercholesterolemic tetrazol-1-yl intermediates BRISTOL-MYERS COMPANY (US) 1991-04-23 US disclosed
EP-0355820-A1 Antihypercholesterolemic tetrazol-1-yl compounds Bristol-Myers Squibb Company (US) 1990-02-28 EP disclosed
US-4870187-A ANTILIPEMIC, ATHEROSCLEROSIS BRISTOL-MYERS COMPANY (US) 1989-09-26 US disclosed