SCHEMBL9788668

SCHEMBL9788668

Cc1ccc2nc(-c3ccc([N+](=O)[O-])cc3)c(CN(C)C(=O)CC(C)C)n2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.54
GABRB2 P47870 5/20 0.54
KDM4E B2RXH2 1/20 0.54
LMNA P02545 1/20 0.54
ALB P02768 1/20 0.54
CYP3A4 P08684 1/20 0.54
CHRM1 P11229 1/20 0.54
HPGD P15428 1/20 0.54
GABRB1 P18505 1/20 0.54
GABRG2 P18507 1/20 0.54
GABRB3 P28472 1/20 0.54
GABRA3 P34903 1/20 0.54
ADRA1A P35348 1/20 0.54
OPRK1 P41145 1/20 0.54
HTR2B P41595 1/20 0.54
GABRA2 P47869 1/20 0.54
KCNH2 Q12809 1/20 0.54
HSD17B10 Q99714 1/20 0.54
TSPO P30536 2/20 0.50
ALOX5 P09917 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10467217 0.94 TSPO (0.55) GABRA1GABRB2KDM4ELMNAALB
SCHEMBL10385117 0.90 GABRA1 (0.66) GABRA1GABRB2KDM4ELMNAALB
SCHEMBL9788699 0.86 GABRA1 (0.58) GABRA1GABRB2KDM4ELMNAALB
SCHEMBL4260189 0.85 GABRA1 (0.55) GABRA1GABRB2KDM4ELMNAALB
Necopidem SCHEMBL1061121 0.85 GABRA1 (0.57) GABRA1GABRB2KDM4ELMNAALB
Hydrochloric Acid SCHEMBL10384385 0.85 GABRB2 (0.57) GABRA1GABRB2KDM4ELMNAALB
SCHEMBL9788663 0.83 GABRA1 (0.55) GABRA1GABRB2KDM4ELMNAALB
SCHEMBL10467508 0.83 GABRA1 (0.55) GABRA1GABRB2KDM4ELMNAALB
SCHEMBL10761650 0.83 GABRA1 (0.54) GABRA1GABRB2KDM4ELMNAALB
SCHEMBL10468528 0.83 ALOX5 (0.49) GABRA1GABRB2KDM4ELMNAALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990506-A Sedatives, anxiolytic, antiulcer, antistress SYNTHELABO (FR) 1991-02-05 US disclosed
US-4891371-A HYPNOTIC, ANXIOLYTIC, ANTI-STRESS ULCER SYNTHELABO (FR) 1990-01-02 US disclosed