SCHEMBL9803467

SCHEMBL9803467

COc1ccc(C(N)=C2C(=O)CCCC2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.50
CA2 P00918 4/20 0.50
PARP10 Q53GL7 2/20 0.50
PARP1 P09874 1/20 0.50
PARP2 Q9UGN5 1/20 0.50
PARP4 Q9UKK3 1/20 0.50
MAPT P10636 4/20 0.48
KDM4E B2RXH2 3/20 0.48
CYP1A2 P05177 2/20 0.48
MEN1 O00255 1/20 0.48
CYP2D6 P10635 1/20 0.48
THRB P10828 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
RECQL P46063 1/20 0.48
BLM P54132 1/20 0.48
KMT2A Q03164 1/20 0.48
HPGD P15428 3/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9802774 0.81 HPD (0.41) MAPTCYP1A2MEN1CYP2D6CYP2C19
SCHEMBL4292937 0.70 ALDH1A1 (0.50) CA1CA2PARP10PARP1PARP2
SCHEMBL4284446 0.69 HPGD (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL201761 0.68 PARP10 (1.00) CA1CA2PARP10PARP1PARP2
SCHEMBL10925317 0.67 CA1 (0.67) CA1CA2PARP10PARP1PARP2
SCHEMBL13207340 0.67 TDP1 (0.75) MAPTCYP1A2CYP2C9CYP2C19BLM
Hydrochloric Acid SCHEMBL408766 0.66 PARP10 (0.95) CA1CA2PARP10PARP1PARP2
Hydrochloric Acid SCHEMBL4376056 0.66 PARP10 (0.95) CA1CA2PARP10PARP1PARP2
SCHEMBL16936986 0.66 MAOA (0.55) CA1CA2MAPTKDM4ECYP1A2
SCHEMBL15708391 0.65 CA1 (0.69) CA1CA2PARP10PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068334-A Analgesics and antipyretics KARL THOMAE GMBH (DE) 1991-11-26 US disclosed
EP-0338228-A2 Use of quinoline-2,5-diones in a medicament having an analgesic, antipyretic and/or antiphlogistic activity Dr. Karl Thomae GmbH (DE) 1989-10-25 EP disclosed