SCHEMBL980380

SCHEMBL980380

O=C(Nc1cccc(N2CCOCC2)c1)c1cc2cccc(O)c2oc1=O

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SETD2 Q9BYW2 1/20 0.52
BACE1 P56817 2/20 0.51
PKM P14618 1/20 0.51
AKR1C3 P42330 7/20 0.50
MAOA P21397 2/20 0.50
MAOB P27338 1/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HCRTR1 O43613 1/20 0.48
CBR1 P16152 3/20 0.48
AR P10275 2/20 0.48
POLB P06746 1/20 0.48
KIF18A Q8NI77 1/20 0.47
SCN10A Q9Y5Y9 1/20 0.47
RPS6KA2 Q15349 1/20 0.47
CASP3 P42574 1/20 0.46
CASP7 P55210 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL981240 0.87 BACE1 (0.68) BACE1PKMMEN1KMT2AHCRTR1
SCHEMBL18132587 0.75 KMO (0.56) SETD2MEN1KMT2AKIF18ACASP3
SCHEMBL979968 0.74 GAPDH (0.53) AKR1C3MAOAMAOBMEN1KMT2A
SCHEMBL6424561 0.74 KMO (0.63) SETD2PKMPOLBRPS6KA2
SCHEMBL979803 0.73 MAOB (0.51) AKR1C3MAOAMAOBKMT2ACBR1
SCHEMBL982797 0.73 AKR1C3 (0.59) AKR1C3MAOAMAOBCBR1AR
SCHEMBL980671 0.73 MAPK1 (0.55) AKR1C3MAOAMAOBCBR1AR
SCHEMBL16583818 0.73 KMO (0.61) SETD2MEN1KMT2AHCRTR1POLB
SCHEMBL981025 0.73 CASP3 (0.51) AKR1C3MAOAMAOBKMT2ACBR1
SCHEMBL978163 0.72 MAOB (0.52) AKR1C3MAOAMAOBCBR1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110021522-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021522-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 CASP7, CASP3, CASP6 SETD2 3827/4885BACE1 76/4885PKM 3415/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.