SCHEMBL9811540

SCHEMBL9811540

O=P(O)(O)C(O)(CCN1CCC(c2cccs2)CC1)P(=O)(O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
MAP1LC3B Q9GZQ8 3/20 0.40
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
KDM4A O75164 1/20 0.36
KDM4B O94953 1/20 0.36
KDM5C P41229 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
KDM3A Q9Y4C1 1/20 0.36
GAA P10253 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9298267 0.80 SLC18A3 (0.57) KMT2ATSHRDRD2SLC18A3MEN1
SCHEMBL9811419 0.79 CCR2 (0.40) DRD2SLC18A3FDPSKCNA3
SCHEMBL9811461 0.78 HRH3 (0.46) DRD2SLC18A3FDPSKCNA3
SCHEMBL9811498 0.76 ALDH1A1 (0.53) ALDH1A1MAPTKMT2ALMNATSHR
SCHEMBL6221175 0.75 SLC18A3 (0.55) KMT2ATSHRCHRM2CHRM4CHRM5
SCHEMBL6223991 0.75 DRD2 (0.57) KMT2ADRD2DRD4DRD3MEN1
SCHEMBL9811433 0.75 DRD2 (0.46) DRD2DRD4DRD3SLC18A3KCNA3
SCHEMBL9811522 0.75 DRD2 (0.48) DRD2DRD3SLC18A3
SCHEMBL9811541 0.75 DRD4 (0.50) ALDH1A1DRD2DRD4DRD3FDPS
SCHEMBL9811477 0.74 FDPS (0.49) ALDH1A1MAPTLMNASLC18A3FDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0272208-B1 AROMATICALLY SUBSTITUTED AZACYCLO-ALKYLALKANEDIPHOSPHONIC ACIDS CIBA-GEIGY AG (CH) 1991-06-12 EP disclosed
US-4871720-A Aromatically substituted azacycloalkyl-alkanediphosphonic acids useful for the treatment of illnesses that can be attributed to calcium metabolism disorders CIBA-GEIGY CORPORATION (US) 1989-10-03 US disclosed
EP-0272208-A1 Aromatically substituted azacyclo-alkylalkanediphosphonic acids CIBA-GEIGY AG (CH) 1988-06-22 EP disclosed