SCHEMBL9815440

SCHEMBL9815440

[CH2]Cc1c(C)n(C(=O)/C=C/c2ccccc2)c2ccc(OC)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2D6 P10635 2/20 0.53
CYP2C9 P11712 2/20 0.53
HIF1A Q16665 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
TSHR P16473 1/20 0.53
NFKB1 P19838 1/20 0.53
PLA2G2A P14555 2/20 0.52
AKR1C3 P42330 8/20 0.49
AKR1C2 P52895 7/20 0.49
ALOX5 P09917 2/20 0.48
PTGS2 P35354 2/20 0.46
CNR1 P21554 2/20 0.46
CNR2 P34972 2/20 0.46
PPARG P37231 2/20 0.46
KDM4E B2RXH2 2/20 0.46
AKR1C4 P17516 2/20 0.46
PTGS1 P23219 2/20 0.46
AKR1C1 Q04828 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9815439 1.00 LMNA (0.53) LMNACYP1A2CYP2D6CYP2C9HIF1A
Cinmetacin SCHEMBL29974302 0.89 LMNA (0.68) LMNACYP1A2CYP2D6CYP2C9HIF1A
Cinmetacin SCHEMBL25138 0.89 LMNA (0.68) LMNACYP1A2CYP2D6CYP2C9HIF1A
Cinmetacin SCHEMBL25139 0.89 LMNA (0.68) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL13229808 0.88 LMNA (0.53) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL12609001 0.88 LMNA (0.58) LMNACYP1A2CYP2D6CYP2C9HIF1A
Cinmetacin SCHEMBL8636225 0.88 LMNA (0.67) LMNACYP1A2CYP2D6CYP2C9HIF1A
Cinmetacin SCHEMBL8636226 0.88 LMNA (0.67) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL12628642 0.88 AKR1C3 (0.62) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL3459041 0.88 PLA2G2A (0.69) LMNACYP1A2CYP2D6CYP2C9HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0452908-A2 Lipoxygenase-inhibiting compounds derived from non-steroidal antiinflammatory carboxylic acids ABBOTT LABORATORIES (US) 1991-10-23 EP disclosed