Cinmetacin

Cinmetacin

SCHEMBL25139

COc1ccc2c(c1)c(CC(=O)O)c(C)n2C(=O)C=Cc1ccccc1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.68
CYP1A2 P05177 4/20 0.68
CYP2C9 P11712 4/20 0.68
HIF1A Q16665 3/20 0.68
NPSR1 Q6W5P4 3/20 0.68
TSHR P16473 3/20 0.68
CYP2D6 P10635 2/20 0.68
NFKB1 P19838 2/20 0.68
AKR1C3 P42330 8/20 0.63
AKR1C2 P52895 7/20 0.63
PLA2G2A P14555 2/20 0.59
PLA2G1B P04054 1/20 0.59
PMP22 Q01453 3/20 0.59
AKR1C4 P17516 2/20 0.59
AKR1C1 Q04828 2/20 0.59
MEN1 O00255 2/20 0.59
MAPT P10636 2/20 0.59
KMT2A Q03164 2/20 0.59
KDM4E B2RXH2 2/20 0.59
PTGS2 P35354 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cinmetacin SCHEMBL25138 1.00 LMNA (0.68) LMNACYP1A2CYP2C9HIF1ANPSR1
Cinmetacin SCHEMBL29974302 1.00 LMNA (0.68) LMNACYP1A2CYP2C9HIF1ANPSR1
Cinmetacin SCHEMBL8636226 0.99 LMNA (0.67) LMNACYP1A2CYP2C9HIF1ANPSR1
Cinmetacin SCHEMBL8636225 0.99 LMNA (0.67) LMNACYP1A2CYP2C9HIF1ANPSR1
SCHEMBL12609001 0.93 LMNA (0.58) LMNACYP1A2CYP2C9HIF1ANPSR1
SCHEMBL3459041 0.92 PLA2G2A (0.69) LMNACYP1A2CYP2C9HIF1ANPSR1
SCHEMBL12628642 0.92 AKR1C3 (0.62) LMNACYP1A2CYP2C9HIF1ANPSR1
SCHEMBL13849829 0.91 PTGS2 (0.61) LMNACYP1A2CYP2C9HIF1ANPSR1
SCHEMBL9815440 0.89 LMNA (0.53) LMNACYP1A2CYP2C9HIF1ANPSR1
SCHEMBL9815439 0.89 LMNA (0.53) LMNACYP1A2CYP2C9HIF1ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4394 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4470565-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT OnQuality Pharmaceuticals China Ltd. (CN) 2024-12-04 EP claimed
US-RE50218-E1 Non-steroidal anti-inflammatory ophthalmic compositions SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2024-11-26 US claimed
CN-118742325-A Methods for preventing or treating diseases or conditions associated with antineoplastic agents 上海岸阔医药科技有限公司 2024-10-01 CN claimed
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
EP-3752201-B1 SUSPENSION OF NANOSCALE, ORGANIC PARTICLES AND PROCESS FOR PRODUCTION THEREOF UNIV FRIEDRICH ALEXANDER ER (DE) 2023-11-22 EP claimed
WO-2023142996-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT 上海岸阔医药科技有限公司 2023-08-03 WO claimed
EP-4034087-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS Research Inc. (CA) 2022-08-03 EP claimed
US-20220218611-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS RESEARCH INC. (CA) 2022-07-14 US claimed
EP-3998932-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS Parsons, C. Lowell (US) 2022-05-25 EP claimed
US-20210145763-A1 LOW THC HEMP EXTRACT AND METHOD OF TREATMENT OR PREVENTION OF AN EYE DISEASE EYE CO PTY LTD. (AU) 2021-05-20 US claimed
EP-0173729-B1 PROCESS FOR SOLUBILIZING ACTIVE PRINCIPLES AND PHARMACEUTICAL COMPOSITIONS THUS OBTAINED CORBIERE, Jérôme (FR) 1990-10-17 EP claimed
EP-0374602-A1 Lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1990-06-27 EP claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
US-4376767-A ANTIBIOTICS AND PHARMACEUTICALS MERCK & CO., INC. (US) 1983-03-15 US claimed
EP-0055870-A1 Pyridylmethyl esters of selected bio-affecting carboxylic acids, process for preparing and pharmaceutical composition comprising the same MERCK & CO. INC. (US) 1982-07-14 EP claimed
EP-0051278-A1 Soft tertiary amine esters of bio-affecting carboxylic acids, processes for preparing and a pharmaceutical composition containing the same MERCK & CO. INC. (US) 1982-05-12 EP claimed
US-4309420-A Stable injectable solutions of indoleacetic acid derivatives A. NATTERMANN & CIE. GMBH (DE) 1982-01-05 US claimed
US-4247554-A ADMINISTERING A QUINAZOLINONE COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1981-01-27 US claimed
US-4083981-A INDOLE-3-ACETIC ACID DERIVATIVES AND NARCOTIC SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1978-04-11 US claimed
US-4029798-A SYNERGISTIC MIXTURE OF INDOLE-3-ACETIC ACID DERIVATIVE AND NARCOTIC SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1977-06-14 US claimed