SCHEMBL9818927

SCHEMBL9818927

N#Cc1ccc(NC(=O)C(C#N)C(=O)c2ccc(C(F)(F)F)cc2)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.48
RAPGEF3 O95398 6/20 0.45
RAPGEF4 Q8WZA2 4/20 0.42
S1PR3 Q99500 1/20 0.41
AR P10275 2/20 0.40
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
KCNE1 P15382 1/20 0.40
KCNQ1 P51787 1/20 0.40
SLC22A12 Q96S37 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN6 P29350 1/20 0.40
PTPN11 Q06124 1/20 0.40
BLM P54132 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819335 0.90 IDO1 (0.50) IDO1RAPGEF3RAPGEF4KCNQ3KCNQ2
SCHEMBL9818996 0.88 IDO1 (0.46) IDO1S1PR3BLM
SCHEMBL9818928 0.85 EPHX2 (0.50) IDO1RAPGEF3RAPGEF4KCNQ3KCNQ2
SCHEMBL9818823 0.84 RHOC (0.49) IDO1RAPGEF3RAPGEF4KCNQ3KCNQ2
SCHEMBL9819165 0.84 RHOC (0.49) IDO1RAPGEF3RAPGEF4KCNQ3KCNQ2
SCHEMBL9819414 0.83 LMNA (0.45) IDO1RAPGEF3RAPGEF4ARKCNQ3
SCHEMBL9819209 0.83 IDO1 (0.47) IDO1RAPGEF3RAPGEF4KCNQ3KCNQ2
SCHEMBL9819035 0.82 MLYCD (0.52)
SCHEMBL9819032 0.82 MLYCD (0.52)
SCHEMBL9819042 0.81 MAOB (0.47) RAPGEF3RAPGEF4PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed