SCHEMBL9828735

SCHEMBL9828735

CCN1C(C)=C(OC(=O)OC(C)C)C(c2sccc2C)C2=C1COC2=O

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PYGM P11217 3/20 0.33
PYGL P06737 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828158 0.91 PYGM (0.35) PYGMPYGL
SCHEMBL9829012 0.88 KDM4E (0.33) KDM4ECYP1A2CYP3A4GAAMAPT
SCHEMBL10425201 0.86 PYGM (0.45) KDM4ECYP1A2CYP3A4GAAMAPT
SCHEMBL9827653 0.86 PYGM (0.35) PYGMPYGL
SCHEMBL10968852 0.84 PYGM (0.37) KDM4EGAAPYGMPYGL
SCHEMBL9829022 0.81 PYGL (0.48) PYGMPYGL
SCHEMBL10969370 0.79 PYGM (0.35) KDM4EPYGMPYGL
SCHEMBL10424875 0.78 PYGM (0.46) PYGMPYGL
SCHEMBL10374452 0.76 PYGM (0.36) PYGMPYGL
SCHEMBL10426101 0.76 ADORA2B (0.42) KDM4ECYP1A2CYP3A4GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0229963-B1 4-THIENYL-DIHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICAL PREPARATIONS BAYER AG (DE) 1991-09-11 EP disclosed
EP-0229963-A2 4-Thienyl-dihydropyridines, process for their preparation and their use as pharmaceutical preparations BAYER AG (DE) 1987-07-29 EP disclosed