SCHEMBL9829012

SCHEMBL9829012

CC1=C(OC(=O)OC(C)C)C(c2sccc2C)C2=C(COC2=O)N1C

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
ADORA2B P29275 2/20 0.32
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828735 0.88 KDM4E (0.36) KDM4ECYP1A2CYP3A4GAAMAPT
SCHEMBL10426101 0.85 ADORA2B (0.42) KDM4ECYP1A2CYP3A4GAAMAPT
SCHEMBL9828158 0.79 PYGM (0.35)
SCHEMBL9045462 0.79 SLC6A3 (0.38) CYP1A2CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL10425201 0.76 PYGM (0.45) KDM4ECYP1A2CYP3A4GAAMAPT
SCHEMBL9827653 0.74 PYGM (0.35)
SCHEMBL10968852 0.72 PYGM (0.37) KDM4EGAATSHRHSD17B10
SCHEMBL9830677 0.71 ALDH1A1 (0.41) KDM4ECYP1A2CYP3A4GAAMAPT
SCHEMBL10424603 0.69 HSD17B10 (0.56) KDM4ECYP1A2CYP3A4GAAMAPT
SCHEMBL9829022 0.69 PYGL (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0229963-B1 4-THIENYL-DIHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICAL PREPARATIONS BAYER AG (DE) 1991-09-11 EP disclosed
EP-0229963-A2 4-Thienyl-dihydropyridines, process for their preparation and their use as pharmaceutical preparations BAYER AG (DE) 1987-07-29 EP disclosed