SCHEMBL9829856

SCHEMBL9829856

Cc1cc(S(N)(=O)=O)sc1S(=O)(=O)c1cccc(CN(C)C)c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 15/20 0.48
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
TSHR P16473 1/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
THRB P10828 1/20 0.33
G6PD P11413 1/20 0.33
PABPC1 P11940 1/20 0.33
KMT2A Q03164 1/20 0.33
HKDC1 Q2TB90 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SLC6A4 P31645 2/20 0.32
SLC6A2 P23975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829067 0.81 CA2 (0.70) CA2MAPTKDM4EMEN1ALDH1A1
SCHEMBL9828452 0.69 CA2 (0.54) CA2CA12CA1CA9ALDH1A1
SCHEMBL9828431 0.66 CA2 (0.64) CA2MAPTKDM4EMEN1ALDH1A1
SCHEMBL3363463 0.66 CA2 (0.45) CA2CA12CA1CA9TSHR
SCHEMBL8045011 0.65 ALDH1A1 (0.52) TSHRMAPTKDM4EMEN1ALDH1A1
SCHEMBL9827904 0.65 CA2 (1.00) CA2MAPTKDM4EMEN1ALDH1A1
SCHEMBL1698715 0.65 GABRA1 (0.54) TSHRMAPTKDM4EMEN1ALDH1A1
Hydrochloric Acid SCHEMBL29426319 0.64 CA2 (0.97) CA2MAPTKDM4EMEN1ALDH1A1
SCHEMBL9068633 0.64 ALDH1A1 (0.52) CA2CA1MAPTKDM4EMEN1
SCHEMBL10388063 0.63 CA2 (0.54) CA2CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295049-B1 THIOPHENE SULFONAMIDE ANTIGLAUCOMA AGENTS MERCK & CO. INC. (US) 1991-10-09 EP disclosed
US-4847289-A Thiophene sulfonamide antiglaucoma agents MERCK & CO., INC. (US) 1989-07-11 US disclosed
EP-0295049-A2 Thiophene sulfonamide antiglaucoma agents MERCK & CO. INC. (US) 1988-12-14 EP disclosed