SCHEMBL9829970

SCHEMBL9829970

N#CC(C#N)=C1CCN(C2CCCC2)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 1/20 0.35
HIF1A Q16665 1/20 0.35
HRH3 Q9Y5N1 3/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
MEN1 O00255 2/20 0.31
USP2 O75604 2/20 0.31
LMNA P02545 2/20 0.31
POLB P06746 2/20 0.31
MAPT P10636 2/20 0.31
HTT P42858 2/20 0.31
RECQL P46063 2/20 0.31
KMT2A Q03164 2/20 0.31
MAPK1 P28482 1/20 0.31
BLM P54132 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10408223 0.98 ALDH1A1 (0.37) ALDH1A1KDM4EHIF1AHRH3DRD2
SCHEMBL9832753 0.93 DRD2 (0.34) DRD2DRD3
SCHEMBL10407364 0.70 CHRM5 (0.43) ALDH1A1HRH3OPRM1SMN1; SMN2HSD17B10
SCHEMBL9829972 0.68 DRD2 (0.36) ALDH1A1HRH3DRD2DRD3MEN1
SCHEMBL9830062 0.67 ALDH1A1 (0.35) ALDH1A1HRH3DRD2DRD3MEN1
SCHEMBL9830847 0.65 OPRM1 (0.41) HRH3OPRM1OPRK1MAPK1KCNH2
SCHEMBL9832183 0.64 NOS3 (0.36) ALDH1A1HRH3MEN1USP2LMNA
SCHEMBL21047873 0.63 OPRM1 (0.43) OPRM1OPRK1MEN1KMT2AMAPK1
SCHEMBL21047698 0.63 OPRM1 (0.43) OPRM1OPRK1MEN1KMT2AMAPK1
SCHEMBL21047786 0.63 OPRM1 (0.43) OPRM1OPRK1MEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed
US-4925939-A 6,7-dihydropyrrol[3,4-c]pyrido[2,3-d]pyrimidine derivatives SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-05-15 US disclosed