SCHEMBL9832290

SCHEMBL9832290

COc1ccc(CN2CCC(=C(C#N)C#N)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.50
ABCC1 P33527 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.50
SIGMAR1 Q99720 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.48
TNF P01375 1/20 0.45
NOD2 Q9HC29 1/20 0.45
NOD1 Q9Y239 1/20 0.45
PTGIR P43119 1/20 0.45
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
COMT P21964 1/20 0.44
KDM4E B2RXH2 1/20 0.43
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
DHFR P00374 1/20 0.42
POLB P06746 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832337 0.86 KMT2A (0.43) ABCB1ABCC1ABCG2SIGMAR1KDM4E
SCHEMBL9832675 0.85 SIGMAR1 (0.54) SIGMAR1DRD4KDM4EMEN1KMT2A
SCHEMBL9832990 0.85 ALDH1A1 (0.45) SMN1; SMN2NOD1KDM4EPOLBMEN1
SCHEMBL10408096 0.83 KDM4E (0.53) ABCB1ABCC1ABCG2KDM4EMEN1
SCHEMBL9832661 0.81 KMT2A (0.52) SIGMAR1KDM4EUSP2MEN1KMT2A
SCHEMBL9831029 0.81 KDM4E (0.60) ABCB1SMN1; SMN2KDM4ETSHRPOLB
SCHEMBL9830403 0.81 MAPT (0.48) KDM4ETSHRPOLBMEN1KMT2A
SCHEMBL9831681 0.76 MEN1 (0.49) SIGMAR1COMTKDM4EUSP2TSHR
SCHEMBL9831145 0.76 HTR3E (0.44) SIGMAR1SMN1; SMN2DRD2TSHRPOLB
SCHEMBL3690085 0.75 PTGIR (0.54) ABCB1ABCC1ABCG2SIGMAR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed
US-4925939-A 6,7-dihydropyrrol[3,4-c]pyrido[2,3-d]pyrimidine derivatives SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-05-15 US disclosed