SCHEMBL9832675

SCHEMBL9832675

COc1cccc(CN2CCC(=C(C#N)C#N)C2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.54
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 4/20 0.52
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.48
CHRM2 P08172 1/20 0.48
HTR1A P08908 1/20 0.48
CHRM3 P20309 1/20 0.48
DRD4 P21917 1/20 0.48
ADRA1D P25100 1/20 0.48
HTR2C P28335 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
DRD3 P35462 1/20 0.48
HTR2B P41595 1/20 0.48
SLC6A3 Q01959 1/20 0.48
TMEM97 Q5BJF2 1/20 0.48
GAA P10253 1/20 0.47
MAPT P10636 2/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832337 0.87 KMT2A (0.43) SIGMAR1KDM4EKMT2AMEN1GAA
SCHEMBL9832290 0.85 ABCB1 (0.50) SIGMAR1KDM4EKMT2AMEN1DRD4
SCHEMBL9830298 0.84 ALDH1A1 (0.45) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL10408096 0.81 KDM4E (0.53) KDM4EALDH1A1KMT2AMEN1GAA
SCHEMBL9832661 0.80 KMT2A (0.52) SIGMAR1KDM4EALDH1A1KMT2AMEN1
SCHEMBL9830403 0.80 MAPT (0.48) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL9831029 0.80 KDM4E (0.60) KDM4EALDH1A1KMT2AMEN1GAA
SCHEMBL10407107 0.78 CA9 (0.56) KDM4EALDH1A1KMT2AMEN1GAA
SCHEMBL10408045 0.77 ADRB1 (0.48) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL667489 0.77 SIGMAR1 (0.62) SIGMAR1KDM4EALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed
US-4925939-A 6,7-dihydropyrrol[3,4-c]pyrido[2,3-d]pyrimidine derivatives SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-05-15 US disclosed