SCHEMBL9834649

SCHEMBL9834649

C=CCC1C(=O)Nc2cc3c(cc21)NC(C)N3

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
PGR P06401 1/20 0.32
MAPT P10636 2/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32
KDM4E B2RXH2 1/20 0.31
GLA P06280 1/20 0.31
HTT P42858 1/20 0.31
NQO2 P16083 3/20 0.31
BRPF1 P55201 1/20 0.30
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833215 0.80 ALDH1A1 (0.41) ALDH1A1PGRKDM4E
SCHEMBL9833705 0.79 PGR (0.41) ALDH1A1PGRMAPTTP53POLB
SCHEMBL9832316 0.78 ALDH1A1 (0.47) ALDH1A1PGRMAPTTP53POLB
SCHEMBL9834636 0.78 ALDH1A1 (0.37) ALDH1A1PGR
SCHEMBL9834483 0.77 IDO1 (0.35) PGRMAPTTP53POLBNQO2
SCHEMBL9835978 0.75 PGR (0.43) PGRTP53POLBBRPF1CREBBP
SCHEMBL9834640 0.72 CHRNB2 (0.39) ALDH1A1MAPTTP53POLBKDM4E
SCHEMBL1455790 0.71 IDO1 (0.58) ALDH1A1MAPTKDM4EBRPF1CREBBP
SCHEMBL9835029 0.70 MAOB (0.39) MAPTTP53BRPF1CREBBP
SCHEMBL9833436 0.70 BRPF1 (0.30) BRPF1CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed