SCHEMBL9836649

SCHEMBL9836649

CN1C(=O)C2=C(c3cccc(C#N)c3)N(C)C(=O)C2=C1c1cccc(C#N)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.46
BRD4 O60885 1/20 0.45
TGFBR1 P36897 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
BACE1 P56817 6/20 0.43
XDH P47989 1/20 0.43
SLC22A12 Q96S37 1/20 0.43
CASP3 P42574 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
CHEK1 O14757 1/20 0.43
CTSD P07339 3/20 0.42
BACE2 Q9Y5Z0 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25028116 0.79 F11 (0.43) PGRBRD4CLK4XDHSLC22A12
SCHEMBL9837439 0.76 RAB9A (0.41) PGRTGFBR1CLK4
SCHEMBL6003407 0.75 BRD4 (0.43) PGRBRD4TGFBR1CLK4BACE1
SCHEMBL9834685 0.75 PGR (0.51) PGRTGFBR1BACE1
SCHEMBL25027823 0.73 SMO (0.46) BRD4CLK4XDHSLC22A12
SCHEMBL2154026 0.72 CLK4 (0.65) PGRCLK4XDHSLC22A12
SCHEMBL11555464 0.71 BRD4 (0.54) PGRBRD4TGFBR1CLK4BACE1
SCHEMBL27787243 0.70 CLK4 (0.63) PGRCLK4XDHSLC22A12
SCHEMBL14620062 0.70 COMT (0.40) BRD4BACE1
SCHEMBL21189130 0.69 CLK4 (0.57) PGRCLK4XDHSLC22A12CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0133156-B1 1,4-DIKETOPYRROLO-(3,4-C) PYRROLES CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
US-4666455-A Compositions pigmented with N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1987-05-19 US disclosed
US-4585878-A N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1986-04-29 US disclosed
EP-0133156-A2 1,4-Diketopyrrolo-(3,4-c) pyrroles CIBA-GEIGY AG (CH) 1985-02-13 EP disclosed