SCHEMBL983765

SCHEMBL983765

CCCCc1c(O)cccc1C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.48
TRIM24 O15164 1/20 0.47
TRIM33 Q9UPN9 1/20 0.47
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
IAPP P10997 3/20 0.45
HTT P42858 2/20 0.42
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
BID P55957 3/20 0.40
MCL1 Q07820 3/20 0.40
BCL2L1 Q07817 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7249953 0.95 ERN1 (0.47) ERN1TRIM24TRIM33CA1CA2
SCHEMBL29210937 0.93 BID (0.48) ERN1TRIM24TRIM33CA1CA2
SCHEMBL6893190 0.89 ERN1 (0.52) ERN1TRIM24TRIM33CA1CA2
SCHEMBL9627639 0.83 IAPP (0.42) IAPPHTTNPC1HPGDMAPK1
SCHEMBL986041 0.82 ERN1 (0.55) ERN1TRIM24TRIM33CA1CA2
SCHEMBL70772 0.81 HTT (0.59) IAPPHTTNPC1HPGDMAPK1
SCHEMBL27464370 0.81 LIPG (0.40) ALDH1A1MEN1MAPTKMT2ABID
SCHEMBL7397839 0.80 TRIM24 (0.48) ERN1TRIM24TRIM33CA1CA2
SCHEMBL23829701 0.79 HPGD (0.42) ERN1IAPPHTTNPC1HPGD
SCHEMBL11452728 0.79 ALDH1A1 (0.38) ERN1CA1CA2IAPPHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1589136-A Pharmaceutical and cosmetic compositions containing aromatic aldehydes bearing oxygen-containing groups CUTANIX CORP (US) 2005-03-02 CN claimed
US-20030157154-A1 Compositions containing hydroxy aromatic aldehydes and their use in treatments CUTANIX CORPORATION 2003-08-21 US claimed
CN-102666461-B Ring compound, its production method, radiation-ray sensitive composition and corrosion-resisting pattern formation method MITSUBISHI GAS CHEMICAL CO.,INC. (JP) 2015-09-30 CN disclosed
CN-102973417-A Pharmaceutical and cosmetic compositions containing oxy group-bearing aromatic aldehydes CUTANIX CORP 2013-03-20 CN disclosed
CN-102666461-A Cyclic compound, process for production thereof, radiation-sensitive composition, and resist pattern formation method MITSUBISHI GAS CHEMICAL CO 2012-09-12 CN disclosed
US-8044067-B2 Isoquinolines as IGF-1R inhibitors ANALYTECON S.A. (CH) 2011-10-25 US disclosed
EP-1931636-B1 ISOQUINOLINES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2011-04-13 EP disclosed
US-7875631-B2 e.g.1-(3,5-dichlorophenyl)-2-formyl-6-methoxy-1,2,3,4-tetrahydroisoquinoline; to prevent and/or treat cancer and other abnormal cell growth, and metabolic as well as blood vessel proliferate disorders, in which uncontrolled expression of insulin-like growth factor-1 receptor is observed ANALYTECON S.A. (CH) 2011-01-25 US disclosed
CN-100590118-C Novel style heterocyclic compound as insulin-like growth factors first type acceptor inhibitor ANALYTECON SA 2010-02-17 CN disclosed
US-20090099229-A1 Isoquinolines as IGF-1R Inhibitors ANALYTECON S.A (CH) 2009-04-16 US disclosed
EP-1732898-B1 TETRAHYDROISOQUINOLINE- AND TETRAHYDROBENZAZEPINE DERIVATIVES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2008-01-23 EP disclosed
US-20070129399-A1 Tetrahydroisoquinoline-and tetrahydrobenzazepine derivatives as igf-1r inhibitors ANALYTECON S.A. (CH) 2007-06-07 US disclosed
CN-1922147-A Novel style heterocyclic compound as insulin-like growth factors first type acceptor inhibitor ANALYTECON SA (CH) 2007-02-28 CN disclosed
CN-1589136-A Pharmaceutical and cosmetic compositions containing aromatic aldehydes bearing oxygen-containing groups CUTANIX CORP (US) 2005-03-02 CN disclosed
EP-1443915-A1 PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING OXY GROUP-BEARING AROMATIC ALDEHYDES Cutanix Corporation (US) 2004-08-11 EP disclosed
US-20030157154-A1 Compositions containing hydroxy aromatic aldehydes and their use in treatments CUTANIX CORPORATION 2003-08-21 US disclosed
WO-2003043621-A1 PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING OXY GROUP-BEARING AROMATIC ALDEHYDES CUTANIX CORPORATION (US) 2003-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030157154-A1 Compositions containing hydroxy aromatic aldehydes and their use in treatments TYR, HRH1, HRH2 ERN1 4830/4885TRIM24 3252/4885TRIM33 2340/4885
US-20070129399-A1 Tetrahydroisoquinoline-and tetrahydrobenzazepine derivatives as igf-1r inhibitors IGF1R, INSR, GPR119 ERN1 2489/4885TRIM24 1952/4885TRIM33 3715/4885
US-20090099229-A1 Isoquinolines as IGF-1R Inhibitors IGF1R, IGFBP1, IGF2BP1 ERN1 1619/4885TRIM24 623/4885TRIM33 3200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.