SCHEMBL9838734

SCHEMBL9838734

O=C(O)c1ccc2ccc(N3CCNCC3)nc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
CYP3A4 P08684 3/20 0.51
HSD17B10 Q99714 2/20 0.51
HTR3E A5X5Y0 4/20 0.48
HTR3B O95264 4/20 0.48
HTR3A P46098 4/20 0.48
HTR3D Q70Z44 4/20 0.48
HTR3C Q8WXA8 4/20 0.48
ALDH1A1 P00352 4/20 0.48
PMP22 Q01453 2/20 0.48
HTR2C P28335 2/20 0.48
CYP1A2 P05177 2/20 0.48
SLC6A4 P31645 2/20 0.48
USP2 O75604 1/20 0.48
ADRB1 P08588 1/20 0.48
HTR1A P08908 1/20 0.48
MAPK1 P28482 1/20 0.48
HTR7 P34969 1/20 0.48
HTT P42858 1/20 0.48
HTR6 P50406 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27415238 0.80 PRKCA (0.59) KDM4ECYP3A4HSD17B10HTR3EHTR3B
SCHEMBL2421817 0.78 BPTF (0.56) KDM4ECYP3A4HSD17B10HTR3EHTR3B
SCHEMBL12469440 0.75 PRKCA (0.62) KDM4ECYP3A4HSD17B10HTR3EHTR3B
SCHEMBL28506643 0.75 KDM4E (0.67) KDM4EHSD17B10ALDH1A1TDP1LMNA
SCHEMBL2869584 0.73 BPTF (0.50) KDM4ECYP3A4HSD17B10HTR2CHTR2A
SCHEMBL9837631 0.72 HTR3E (0.49) KDM4ECYP3A4HSD17B10HTR3EHTR3B
SCHEMBL30695563 0.72 ADRB1 (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL5338538 0.72 ALDH1A1 (0.54) KDM4ECYP3A4HSD17B10HTR3EHTR3B
SCHEMBL22790262 0.71 HTR3E (0.51) KDM4ECYP3A4HSD17B10HTR3EHTR3B
SCHEMBL8588025 0.71 HTR3E (0.59) KDM4ECYP3A4HSD17B10HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0159174-B1 SUBSTITUTED NAPHTHYRIDINE-, QUINOLINE- AND BENZOXAZINE- CARBOXYLIC ACIDS AS ANTIBACTERIAL AGENTS AND PROCESSES FOR THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1991-10-23 EP disclosed