SCHEMBL9844783

SCHEMBL9844783

COC(=O)c1ccc(CCCc2cn(C)c3nc(N)n(OC(C)C)c(=O)c23)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 10/20 0.39
CYP4A11 Q02928 2/20 0.39
CYP4F2 P78329 1/20 0.38
TLR8 Q9NR97 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
TP53 P04637 1/20 0.34
IDH1 O75874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844790 0.73 EP300 (0.38) EP300CYP4A11CYP4F2TLR8MAPT
SCHEMBL9844770 0.68 EP300 (0.49) EP300CYP4A11CYP4F2CYP1A2CYP3A4
SCHEMBL9844748 0.67 DRD2 (0.39) EP300MAPTTHRB
SCHEMBL9844768 0.67 TBXAS1 (0.39) EP300MAPT
SCHEMBL12176878 0.65 CYP4A11 (0.70) CYP4A11CYP4F2CYP1A2CYP3A4CYP2C9
SCHEMBL8982456 0.62 CYP4A11 (0.48) EP300CYP4A11CYP4F2CYP1A2CYP3A4
SCHEMBL10169575 0.61 CYP4A11 (0.68) CYP4A11CYP4F2CYP1A2CYP3A4CYP2C9
SCHEMBL5733406 0.61 CYP4A11 (0.72) CYP4A11CYP4F2CYP1A2CYP3A4CYP2C9
SCHEMBL13230897 0.61 CYP4A11 (0.72) CYP4A11CYP4F2CYP1A2CYP3A4CYP2C9
SCHEMBL8982447 0.61 CYP4A11 (0.48) EP300CYP4A11CYP4F2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed