Biguanide

Biguanide

SCHEMBL9846419

CCOCC.N.N=C(N)NC(=N)N

nearest known ligand 0.32

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
TSHR P16473 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
CYP2C19 P33261 1/20 0.31
NOS2 P35228 1/20 0.31
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
PRSS3 P35030 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ether SCHEMBL300500 0.80
Biguanide SCHEMBL27671000 0.77 TSHR (0.40) ALDH1A1CYP1A2CYP2D6TSHRNOS3
Biguanide SCHEMBL6050569 0.77 NOS3 (0.39) CYP1A2CYP2D6TSHRNOS3NOS1
Biguanide SCHEMBL28774142 0.77 NOS3 (0.36) CYP1A2CYP2D6TSHRNOS3NOS1
Biguanide SCHEMBL27622487 0.76
Biguanide SCHEMBL29001087 0.73 ALOX15 (0.68) ALDH1A1ALOX15CYP1A2TSHRCYP2C19
Biguanide SCHEMBL27454502 0.73
Biguanide SCHEMBL8039 0.72
Biguanide SCHEMBL18255803 0.72 MAPK1 (0.31) NOS3NOS1NOS2
Biguanide SCHEMBL25340958 0.72 SPHK1 (0.52) ALDH1A1TSHRNOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456093-A2 Biguanide derivatives and biocidal compositions containing them H.B. FULLER LICENSING & FINANCING, INC. (US) 1991-11-13 EP disclosed