SCHEMBL9848757

SCHEMBL9848757

Cc1cc(N(C)N2C(=O)c3ccccc3C2=O)c(=O)[nH]c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
HPGD P15428 6/20 0.35
KDM4E B2RXH2 5/20 0.35
HSD17B10 Q99714 2/20 0.35
BRD4 O60885 2/20 0.35
GAA P10253 2/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
ALDH1A1 P00352 3/20 0.35
CASP3 P42574 1/20 0.34
ATAD2 Q6PL18 1/20 0.33
GALR3 O60755 1/20 0.33
MAPT P10636 3/20 0.32
HTT P42858 2/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9848768 0.83 MEN1 (0.33) KMT2AMEN1HPGDKDM4EHSD17B10
SCHEMBL8727685 0.67 ALDH1A1 (0.45) KMT2AMEN1HPGDGAAALDH1A1
SCHEMBL9848749 0.66 MAPK1 (0.60) KMT2AMEN1HPGDKDM4EHSD17B10
SCHEMBL873778 0.65 CASP3 (0.52) KMT2AMEN1HPGDKDM4EALDH1A1
SCHEMBL15478582 0.65 HSD17B10 (0.56) HPGDKDM4EHSD17B10BRD4GAA
SCHEMBL20979820 0.65 CASP3 (0.50) KMT2AMEN1KDM4EGAAALDH1A1
SCHEMBL7480856 0.62 SLC6A2 (0.45) KMT2AKDM4EMAPTHTTNPC1
SCHEMBL18917449 0.61 ANPEP (0.44) KMT2AMEN1HPGDHSD17B10ALDH1A1
SCHEMBL15181275 0.59 MEN1 (0.47) KMT2AMEN1KDM4EHSD17B10GAA
SCHEMBL25421078 0.58 KMT2A (0.46) KMT2AMEN1HPGDGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462808-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed