SCHEMBL873778

SCHEMBL873778

CN(C)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.52
CDC25B P30305 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 5/20 0.45
ALDH1A1 P00352 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
CES1 P23141 2/20 0.45
HTT P42858 2/20 0.45
HIF1A Q16665 2/20 0.45
TTR P02766 1/20 0.45
POLB P06746 3/20 0.43
LMNA P02545 3/20 0.43
KDM4E B2RXH2 2/20 0.43
RAB9A P51151 2/20 0.43
BLM P54132 2/20 0.43
MAPK1 P28482 2/20 0.43
CES2 O00748 1/20 0.43
APAF1 O14727 1/20 0.43
TERT O14746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6276424 0.81 HEXA (0.57) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL5707657 0.81 CES1 (0.57) CASP3MEN1KMT2AMAPTALDH1A1
SCHEMBL10100428 0.80 TERT (0.47) MEN1KMT2AALDH1A1SMN1; SMN2HTT
SCHEMBL20979820 0.79 CASP3 (0.50) CASP3CDC25BMEN1KMT2AMAPT
SCHEMBL15181275 0.78 MEN1 (0.47) CASP3MEN1KMT2AMAPTALDH1A1
SCHEMBL8727685 0.78 ALDH1A1 (0.45) CASP3MEN1KMT2AMAPTALDH1A1
SCHEMBL27471585 0.78 DPP4 (0.47) MEN1KMT2AALDH1A1POLB
SCHEMBL11036033 0.76 RNASEH1 (0.56) CASP3MEN1KMT2AMAPTALDH1A1
SCHEMBL11711016 0.76 CA12 (0.46) MEN1KMT2AALDH1A1SMN1; SMN2HTT
SCHEMBL11665542 0.75 CA12 (0.43) CASP3CDC25BMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4016663-A1 ELECTRODE MATERIAL FOR THE PRINTING OF POLYMER BATTERIES Evonik Operations GmbH (DE) 2022-06-22 EP disclosed
US-10053452-B2 Crystalline forms of N-(4-((3-(2-amino-4-pyrimidinyl)-2-pyridinyl)oxy)phenyl)-4-(4-methyl-2-thienyl)-1-phthalazinamine salts and uses thereof AMGEN INC. (US) 2018-08-21 US disclosed
US-9889213-B2 Multimodal imaging of fibrin THE GENERAL HOSPITAL CORPORATION (US) 2018-02-13 US disclosed
US-20160304504-A1 CRYSTALLINE FORMS OF N-(4-((3-(2-AMINO-4-PYRIMIDINYL)-2-PYRIDINYL)OXY)PHENYL)-4-(4-METHYL -2-THIENYL)-1-PHTHALAZINAMINE SALTS AND USES THEREOF AMGEN INC. 2016-10-20 US disclosed
US-20160304504-A1 CRYSTALLINE FORMS OF N-(4-((3-(2-AMINO-4-PYRIMIDINYL)-2-PYRIDINYL)OXY)PHENYL)-4-(4-METHYL -2-THIENYL)-1-PHTHALAZINAMINE SALTS AND USES THEREOF AMGEN INC. 2016-10-20 US disclosed
EP-3077392-A1 CRYSTALLINE FORMS OF N-(4-((3-(2-AMINO-4-PYRIMIDINYL) - 2-PYRIDINYL)OXY)PHENYL)-4-(4-METHYL-2-THIENYL)-1 -PHTHALAZINAMINE PHARMACEUTICALLY ACCEPTABLE SALTS AND USES THEREOF Amgen Inc. (US) 2016-10-12 EP disclosed
US-20160199519-A1 Multimodal Imaging of Fibrin THE GENERAL HOSPITAL CORPORATION 2016-07-14 US disclosed
US-9200017-B2 Multimodal imaging of fibrin THE GENERAL HOSPITAL CORPORATION (US) 2015-12-01 US disclosed
WO-2015084649-A1 CRYSTALLINE FORMS OF N-(4-((3-(2-AMINO-4-PYRIMIDINYL) - 2-PYRIDINYL)OXY)PHENYL)-4-(4-METHYL-2-THIENYL)-1 -PHTHALAZINAMINE PHARMACEUTICALLY ACCEPTABLE SALTS AND USES THEREOF AMGEN INC. (US) 2015-06-11 WO disclosed
WO-2015084649-A1 CRYSTALLINE FORMS OF N-(4-((3-(2-AMINO-4-PYRIMIDINYL) - 2-PYRIDINYL)OXY)PHENYL)-4-(4-METHYL-2-THIENYL)-1 -PHTHALAZINAMINE PHARMACEUTICALLY ACCEPTABLE SALTS AND USES THEREOF AMGEN INC. (US) 2015-06-11 WO disclosed
US-20090023758-A1 Macrocyclic Inhibitors of Hepatitis C Virus MEDIVIR AB (SE) 2009-01-22 US disclosed
WO-2008124083-A2 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC. (US) 2008-10-16 WO disclosed
WO-2008106104-A2 ENVIRONMENTALLY SENSITIVE FLUOROPHORES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2008-09-04 WO disclosed
WO-2008023357-A1 HETEROCYCLIC DERIVATIVES BINDING TO THE PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR (PBR) TECHNION RESEARCH AND DEVELOPMENT FOUNDATION LTD. (IL) 2008-02-28 WO disclosed
EP-1037947-B1 CYANINE DYES AMERSHAM PLC (GB) 2003-09-10 EP disclosed
US-6468730-B2 DI- OR TRIHALO-SUBSTITUTED CARBOXY OR SULFONIC ACID STORAGE STABILIZER FUJI PHOTO FILM CO., LTD. (JP) 2002-10-22 US disclosed
US-6348599-B1 CYANINE DYES HAVING OVERALL POSITIVE CHARGE OF +2 TO +6 AND REACTIVE OR FUNCTIONAL GROUP PRESENT WHICH CAN REACT WITH FUNCTIONAL OR REACTIVE GROUP OF TARGET MOLECULE NYCOMED AMERSHAM PLC (GB) 2002-02-19 US disclosed
US-20020015926-A1 IMAGE RECORDING MATERIAL FUJIFILM CORPORATION (JP) 2002-02-07 US disclosed
EP-1037947-A1 CYANINE DYES Nycomed Amersham plc (GB) 2000-09-27 EP disclosed
WO-1999005221-A1 CYANINE DYES NYCOMED AMERSHAM PLC (GB) 1999-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023758-A1 Macrocyclic Inhibitors of Hepatitis C Virus CTRC, NOX3, HAVCR2 CASP3 50/4885CDC25B 1828/4885MEN1 3400/4885
US-20160199519-A1 Multimodal Imaging of Fibrin FGB, F2, SERPINC1 CASP3 1227/4885CDC25B 4650/4885MEN1 605/4885
US-20160304504-A1 CRYSTALLINE FORMS OF N-(4-((3-(2-AMINO-4-PYRIMIDINYL)-2-PYRIDINYL)OXY)PHENYL)-4-(4-METHYL -2-THIENYL)-1-PHTHALAZINAMINE SALTS AND USES THEREOF BCL9, NPM1, MLLT3 CASP3 819/4885CDC25B 228/4885MEN1 220/4885
US-10053452-B2 Crystalline forms of N-(4-((3-(2-amino-4-pyrimidinyl)-2-pyridinyl)oxy)phenyl)-4-(4-methyl-2-thienyl)-1-phthalazinamine salts and uses thereof BCL9, NPM1, MLLT3 CASP3 819/4885CDC25B 228/4885MEN1 220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.