SCHEMBL9849520

SCHEMBL9849520

N#Cc1ccc(-c2cccc(C(F)(F)F)c2)nc1Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.62
KDM1A O60341 3/20 0.56
CTSK P43235 9/20 0.49
KCNH2 Q12809 5/20 0.47
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
THRB P10828 1/20 0.44
CYP2C9 P11712 1/20 0.44
PKM P14618 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
STAT6 P42226 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26199891 0.82 KIF11 (0.46) CTSSCTSKKDM4EALDH1A1MEN1
SCHEMBL9849371 0.78 CTSS (0.51) CTSSKDM1ACTSKKCNH2KDM4E
SCHEMBL1904903 0.77 CYP1A2 (0.53) KDM4EALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL9205171 0.77 CYP11B2 (0.50) CTSSKDM4EALDH1A1MAOB
SCHEMBL9954071 0.77 CTSS (1.00) CTSSKDM1ACTSKKCNH2KDM4E
SCHEMBL3751766 0.75 KDM1A (0.56) CTSSKDM1AKDM4EALDH1A1MEN1
SCHEMBL6837458 0.75 KDM1A (0.70) CTSSKDM1AKDM4EALDH1A1MEN1
SCHEMBL3873916 0.75 CTSK (0.65) CTSSCTSKKCNH2CYP1A2CYP3A4
SCHEMBL12382082 0.75 ALDH1A1 (0.64) CTSSCTSKKDM4EALDH1A1NPSR1
SCHEMBL6236184 0.74 CTSS (0.57) CTSSKDM1ACTSKKCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed