SCHEMBL9851539

SCHEMBL9851539

O=C1c2c(F)cccc2N=C(F)C1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.35
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
PARP1 P09874 2/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
ALOX12 P18054 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL208466 0.69 CA1 (0.44) CA1CA2CA7CA9HTR2C
SCHEMBL28886119 0.66 NOS1 (0.42) MEN1MAPTKMT2A
SCHEMBL8830105 0.64 TTR (0.37) CA1CA2CA7CA9HTR2C
SCHEMBL21277748 0.59 ADORA2B (0.35) BACE1CA1CA2CA7CA9
SCHEMBL28619081 0.57 CA1 (0.40) CA1CA2CA7CA9HTR2C
SCHEMBL8733810 0.57 CA1 (0.43) CA1CA2CA7CA9HTR2C
SCHEMBL10716838 0.56 MAOA (0.52) CA1CA2CA7CA9MEN1
SCHEMBL13487412 0.56 CA1 (0.52) CA1CA2CA7CA9MEN1
SCHEMBL5866470 0.56 CA1 (0.52) CA1CA2CA7CA9MEN1
SCHEMBL3375220 0.55 CA2 (0.46) CA1CA2CA7CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0424802-A2 Tricyclic quinoline antineoplastic agents ABBOTT LABORATORIES (US) 1991-05-02 EP disclosed