SCHEMBL9852060

SCHEMBL9852060

COc1ccc(CN2CCC(NC(=O)c3cc4ccccc4o3)CC2)c(OC)c1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.60
KDM4E B2RXH2 2/20 0.58
ALDH1A1 P00352 2/20 0.58
HPGD P15428 2/20 0.58
HSD17B10 Q99714 2/20 0.58
MCHR1 Q99705 4/20 0.57
KCNH2 Q12809 2/20 0.57
TP53 P04637 1/20 0.57
UTS2R Q9UKP6 1/20 0.55
DRD4 P21917 2/20 0.55
BCHE P06276 1/20 0.55
SIGMAR1 Q99720 2/20 0.54
RAB9A P51151 1/20 0.53
POLB P06746 1/20 0.53
TSHR P16473 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727091 0.88 DRD4 (0.70) ACHEKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9852062 0.86 DRD4 (0.71) ACHEKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9852245 0.81 DRD4 (0.55) ACHEALDH1A1MCHR1DRD4SIGMAR1
SCHEMBL9727131 0.80 MAOB (0.74) ACHEMCHR1KCNH2UTS2RDRD4
Iodide SCHEMBL9852252 0.79 DRD4 (0.59) ACHEKDM4EALDH1A1HPGDHSD17B10
SCHEMBL4917286 0.79 TP53 (0.67) KDM4EALDH1A1HPGDHSD17B10TP53
SCHEMBL9727140 0.79 UTS2R (0.73) ACHEKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6333472 0.78 MCHR1 (0.69) ACHEMCHR1KCNH2DRD4BCHE
SCHEMBL9852064 0.78 MCHR1 (0.66) ACHEKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9727082 0.78 DRD4 (0.64) ACHEKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416581-A1 Substituted N-benzylpiperidine amides G.D. Searle & Co. (US) 1991-03-13 EP claimed