SCHEMBL9857121

SCHEMBL9857121

COc1ccccc1CC(CCN(C)C)c1ccccc1C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
AOC3 Q16853 1/20 0.40
HTR7 P34969 1/20 0.39
CHRM2 P08172 3/20 0.38
CYP2D6 P10635 3/20 0.37
CYP3A4 P08684 2/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
KCNH2 Q12809 2/20 0.37
SLC6A3 Q01959 1/20 0.37
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
ALOX12 P18054 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9856862 0.79 HTR2A (0.49) KDM4EAOC3HTR7CHRM2CYP2D6
SCHEMBL9856602 0.74 CYP2D6 (0.45) ALDH1A1HTR7CYP2D6POLBHTT
SCHEMBL9857222 0.73 HTR2A (0.49) KDM4EALDH1A1CHRM2CYP2D6CYP3A4
SCHEMBL5403632 0.68 HTR7 (0.46) KDM4EALDH1A1HTR7CYP3A4POLB
SCHEMBL9856971 0.67 KDM4E (0.38) KDM4EALDH1A1HTR7SLC6A2SLC6A4
SCHEMBL9856935 0.67 SLC6A2 (0.49) KDM4EHTR7CHRM2CYP2D6SLC6A2
SCHEMBL2937482 0.66 AOC3 (0.73) AOC3HTR7CHRM2KCNH2TAAR1
SCHEMBL9230337 0.66 HTR2A (0.65) KDM4EHTR7CHRM2CYP2D6CYP3A4
SCHEMBL9857031 0.66 PPARG (0.41) ALDH1A1HTR7CYP2D6SLC6A4MAPT
SCHEMBL8129763 0.66 KDM4E (0.82) KDM4EALDH1A1HTR7CYP2D6HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996235-A Selectively inhibiting the uptake of serotonin and norepinephrine ELI LILLY AND COMPANY (US) 1991-02-26 US disclosed