SCHEMBL9864602

SCHEMBL9864602

CSc1sc(S(C)(=O)=O)cc1C#N

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
USP7 Q93009 2/20 0.32
USP47 Q96K76 1/20 0.32
EPAS1 Q99814 1/20 0.30
GRIA4 P48058 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865123 0.86 KEAP1 (0.35) KEAP1NFE2L2USP7USP47GRIA4
SCHEMBL9865352 0.72 KEAP1 (0.36) KEAP1NFE2L2USP7GRIA4
SCHEMBL3716774 0.71 GRIA2 (0.39) GRIA4
SCHEMBL9864348 0.70 PTGS2 (0.33)
SCHEMBL741497 0.69 KEAP1 (0.71) KEAP1NFE2L2USP7USP47GRIA4
SCHEMBL9864443 0.69 USP7 (0.57) KEAP1NFE2L2USP7USP47GRIA4
SCHEMBL742310 0.63 L3MBTL1 (0.50) KEAP1NFE2L2USP7
SCHEMBL9864759 0.58
SCHEMBL13755141 0.58 PTGS2 (0.39) EPAS1
SCHEMBL3816299 0.58 ALDH1A1 (0.44) KEAP1NFE2L2USP7USP47EPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994485-A Seed and soil fungi, bacteria DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1991-02-19 US disclosed
EP-0234622-B1 NEW THIO COMPOUNDS HAVING FUNGICIDAL ACTIVITY DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-06-27 EP disclosed
EP-0234622-A1 New thio compounds having fungicidal activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1987-09-02 EP disclosed