SCHEMBL9865031

SCHEMBL9865031

Cc1[c]c(-c2cc(Cl)ccc2Cl)no1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.40
DUSP3 P51452 1/20 0.40
PTPN11 Q06124 1/20 0.40
NPSR1 Q6W5P4 2/20 0.38
LMNA P02545 1/20 0.38
HTR2B P41595 1/20 0.38
PDE4D Q08499 1/20 0.38
MAPT P10636 4/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
NTSR1 P30989 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
SAE1 Q9UBE0 1/20 0.36
UBA2 Q9UBT2 1/20 0.36
IDO1 P14902 1/20 0.36
GAA P10253 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9873089 0.85 KCNH2 (0.39) PDE4DMEN1KMT2AHSD11B1PDE2A
SCHEMBL9936299 0.84 HSD11B1 (0.36) RAB9AMAPTTP53HSD11B1GPBAR1
SCHEMBL1086652 0.79 PTGS1 (0.47) RAB9ALMNAMAPTALDH1A1HPGD
SCHEMBL3940018 0.75 NR1H4 (0.42) RAB9ANPSR1MAPTMEN1KMT2A
SCHEMBL11593511 0.73 PTGS1 (0.51) RAB9AMAPTALDH1A1MEN1KMT2A
SCHEMBL1326560 0.70 ALDH1A1 (0.44) NPSR1LMNAMAPTALDH1A1KMT2A
SCHEMBL14363632 0.68 RAB9A (0.51) RAB9ADUSP3PTPN11NPSR1HTR2B
SCHEMBL167920 0.66
SCHEMBL440944 0.66 TP53 (0.61) PTPN11LMNAHTR2BPDE4DMAPT
SCHEMBL29364307 0.66 TP53 (0.61) PTPN11LMNAHTR2BPDE4DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011938-A Antimicrobials ELI LILLY AND COMPANY (US) 1991-04-30 US disclosed
US-4940718-A BACTERICIDES ELI LILLY AND COMPANY (US) 1990-07-10 US disclosed
EP-0202046-A1 7-Substituted bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-11-20 EP disclosed