SCHEMBL9873089

SCHEMBL9873089

Cc1[c]c(-c2cc(Cl)ccc2F)no1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.39
HSD11B1 P28845 1/20 0.35
EPHX2 P34913 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
PTGS1 P23219 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32
GABRA4 P48169 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865031 0.85 RAB9A (0.40) HSD11B1GPBAR1MEN1KMT2APDE4D
SCHEMBL1086256 0.78 NPC1 (0.45) GPBAR1PTGS1MEN1KMT2AL3MBTL1
SCHEMBL9936299 0.76 HSD11B1 (0.36) HSD11B1GPBAR1PTGS1PTGS2
SCHEMBL3940018 0.74 NR1H4 (0.42) GPBAR1MEN1KMT2ASMN1; SMN2
SCHEMBL4970805 0.73 CYP17A1 (0.37) MEN1KMT2AGABRA5
SCHEMBL11593511 0.72 PTGS1 (0.51) GPBAR1PTGS1MEN1KMT2ASMN1; SMN2
SCHEMBL1086652 0.71 PTGS1 (0.47) HSD11B1GPBAR1PTGS1KMT2ASMN1; SMN2
SCHEMBL1679666 0.70 LMNA (0.44) GPBAR1MEN1KMT2ASMN1; SMN2
SCHEMBL6004541 0.67 PTGS2 (0.39) GPBAR1PTGS1KMT2ASMN1; SMN2PTGS2
SCHEMBL6126814 0.67 CNR1 (0.34) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011938-A Antimicrobials ELI LILLY AND COMPANY (US) 1991-04-30 US disclosed
US-4940718-A BACTERICIDES ELI LILLY AND COMPANY (US) 1990-07-10 US disclosed
EP-0202046-A1 7-Substituted bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-11-20 EP disclosed