SCHEMBL9867487

SCHEMBL9867487

CCOC(=O)c1oc2c(C(C)(C)C)cc(C(C)(C)C)c(O)c2c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.48
MAPT P10636 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
KDM4E B2RXH2 2/20 0.41
HSD17B10 Q99714 2/20 0.41
NMT2 O60551 5/20 0.41
NMT1 P30419 5/20 0.41
ADRB2 P07550 2/20 0.40
ADRB1 P08588 2/20 0.40
ADRB3 P13945 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MAPK1 P28482 1/20 0.39
ALOX5 P09917 1/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867508 0.82 NPC1 (0.45) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL9868498 0.82 GLRA3 (0.49) L3MBTL1KDM4EHSD17B10SMN1; SMN2ALOX5
SCHEMBL9866663 0.82 ALOX5 (0.47) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL9866325 0.82 RAB9A (0.58) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL9867051 0.80 RAB9A (0.41) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL9868567 0.80 RAB9A (0.59) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL3609288 0.78 RAB9A (0.50) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL10458678 0.72 L3MBTL1 (0.52) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL9739893 0.71 ALOX5 (0.54) RAB9ANPC1MAPTL3MBTL1KDM4E
SCHEMBL9739459 0.71 ALOX5 (0.53) RAB9ANPC1MAPTL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006549-A Antiinflammatory agents MERCK & CO., INC. (US) 1991-04-09 US disclosed
EP-0399773-A1 Novel 7-aroyl-4-hydroxy-3-methyl benzolfurans as dual inhibitors of cyclooxygenase and 5-lipoxygenase MERCK & CO. INC. (US) 1990-11-28 EP disclosed