SCHEMBL9870774

SCHEMBL9870774

CC(=O)Nc1nnc2c3c(c(N4CCOCC4)nn12)CCCC3

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.40
ALDH1A1 P00352 10/20 0.38
TSHR P16473 2/20 0.38
RXFP1 Q9HBX9 3/20 0.38
KDM4E B2RXH2 7/20 0.37
MAPT P10636 4/20 0.37
GAA P10253 3/20 0.37
MAPK1 P28482 2/20 0.37
HPGD P15428 5/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
HTT P42858 2/20 0.35
HSD17B10 Q99714 3/20 0.35
MTOR P42345 2/20 0.35
ALOX15 P16050 1/20 0.34
LMNA P02545 2/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CA P42336 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871084 0.89 APP (0.37) ACHEALDH1A1TSHRKDM4EMAPT
SCHEMBL9871188 0.88 KDM4E (0.37) ALDH1A1TSHRRXFP1KDM4EMAPT
SCHEMBL9870788 0.83 KDM4E (0.42) ALDH1A1TSHRRXFP1KDM4EMAPT
SCHEMBL10963823 0.77 ALDH1A1 (0.40) ALDH1A1TSHRKDM4EMAPTGAA
SCHEMBL9871963 0.77 HTT (0.40) ALDH1A1TSHRKDM4EMAPTGAA
SCHEMBL9872191 0.76 MAPT (0.38) ALDH1A1TSHRKDM4EMAPTGAA
SCHEMBL9871542 0.75 ALDH1A1 (0.39) ALDH1A1TSHRRXFP1KDM4EMAPT
SCHEMBL9870678 0.74 KDM4E (0.39) ALDH1A1TSHRRXFP1KDM4EMAPT
Hydrochloric Acid SCHEMBL9872400 0.74 ALDH1A1 (0.39) ALDH1A1TSHRRXFP1KDM4EMAPT
SCHEMBL8793570 0.73 LMNA (0.45) ALDH1A1TSHRKDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011835-A Substituted triazolopyridazines, pharmaceutical compositions and use MERRELL DOW PHARMACEUTICALS INC. (US) 1991-04-30 US claimed
US-5011835-A Substituted triazolopyridazines, pharmaceutical compositions and use MERRELL DOW PHARMACEUTICALS INC. (US) 1991-04-30 US disclosed