SCHEMBL8793570

SCHEMBL8793570

CCOC(=O)C(=O)Nc1nnc2c3c(c(N4CCCC4)nn12)CCCC3

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.45
ALDH1A1 P00352 8/20 0.34
HPGD P15428 5/20 0.34
MAPT P10636 4/20 0.34
PKM P14618 2/20 0.34
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
KDM4E B2RXH2 4/20 0.33
HSD17B10 Q99714 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
ACACA Q13085 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
GAA P10253 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870642 0.99 LMNA (0.44) LMNAALDH1A1HPGDMAPTPKM
SCHEMBL9870788 0.92 KDM4E (0.42) LMNAALDH1A1HPGDMAPTKDM4E
SCHEMBL9872191 0.88 MAPT (0.38) LMNAALDH1A1HPGDMAPTKDM4E
SCHEMBL9871963 0.82 HTT (0.40) LMNAALDH1A1HPGDMAPTKDM4E
SCHEMBL9871188 0.75 KDM4E (0.37) LMNAALDH1A1HPGDMAPTKDM4E
SCHEMBL9870774 0.73 ACHE (0.40) LMNAALDH1A1HPGDMAPTKDM4E
SCHEMBL9872179 0.71 MAPT (0.33) ALDH1A1HPGDMAPTPKMKDM4E
SCHEMBL8794028 0.71 KMT2A (0.54) LMNAKDM4ENPC1RAB9APOLB
SCHEMBL10964096 0.70 SMN1; SMN2 (0.39) ALDH1A1NPSR1USP2GAAPOLB
SCHEMBL9871763 0.66 ALDH1A1 (0.35) LMNAALDH1A1HPGDMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011835-A Substituted triazolopyridazines, pharmaceutical compositions and use MERRELL DOW PHARMACEUTICALS INC. (US) 1991-04-30 US claimed
EP-0441339-B1 Substituted triazolopyridazines MERRELL PHARMA INC (US) 1997-08-20 EP disclosed
EP-0441339-A1 Substituted triazolopyridazines MERRELL PHARMACEUTICALS INC. (US) 1991-08-14 EP disclosed
US-5011835-A Substituted triazolopyridazines, pharmaceutical compositions and use MERRELL DOW PHARMACEUTICALS INC. (US) 1991-04-30 US disclosed