SCHEMBL9872977

SCHEMBL9872977

Nc1nc2c(s1)CC(CC(=O)N1CCN(c3ccccn3)CC1)CC2

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.59
ALDH1A1 P00352 7/20 0.59
HSD17B10 Q99714 6/20 0.59
DPP4 P27487 1/20 0.48
HPGD P15428 3/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
LMNA P02545 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
MAPK1 P28482 1/20 0.48
CYP2C19 P33261 1/20 0.48
HTT P42858 1/20 0.48
RECQL P46063 2/20 0.47
CASP1 P29466 1/20 0.45
POLB P06746 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
SCN9A Q15858 2/20 0.44
SCN3A Q9NY46 2/20 0.44
SCN5A Q14524 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL9874788 0.99 KDM4E (0.58) KDM4EALDH1A1HSD17B10DPP4HPGD
Water SCHEMBL9874791 0.99 KDM4E (0.58) KDM4EALDH1A1HSD17B10DPP4HPGD
SCHEMBL9873677 0.83 KDM4E (0.47) KDM4EALDH1A1HSD17B10DPP4HPGD
SCHEMBL9873640 0.83 DRD2 (0.47) HSD17B10LMNAMAPK1HTTPOLB
SCHEMBL9871472 0.82 HTR1A (0.53)
SCHEMBL9872326 0.78 LMNA (0.47) HSD17B10LMNAMAPK1HTTPOLB
Water SCHEMBL9874025 0.77 LMNA (0.46) HSD17B10LMNAMAPK1HTTPOLB
Water SCHEMBL9874020 0.77 LMNA (0.46) HSD17B10LMNAMAPK1HTTPOLB
SCHEMBL8296502 0.74 DPP4 (0.47) DPP4SCN9ASCN3ASCN5ASCN4A
SCHEMBL3163995 0.72 KDM4E (0.50) KDM4EALDH1A1HSD17B10DPP4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988699-A Treatment of psychological disorders such as schizophrenia, as antipsychotic agents and hypotensive agents WARNER-LAMBERT COMPANY (US) 1991-01-29 US disclosed