SCHEMBL9877331

SCHEMBL9877331

O=C(O)CCNC(=S)Nc1ccc2cn[nH]c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.69
HPGD P15428 1/20 0.67
ALDH1A1 P00352 13/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2D6 P10635 1/20 0.67
CYP2C9 P11712 1/20 0.67
CYP2C19 P33261 1/20 0.67
HIF1A Q16665 1/20 0.67
PHLPP2 Q6ZVD8 1/20 0.67
HSD17B10 Q99714 1/20 0.67
MAPT P10636 11/20 0.63
KDM4E B2RXH2 11/20 0.63
RAB9A P51151 2/20 0.63
GAA P10253 2/20 0.63
NPC1 O15118 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
QPCT Q16769 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9877025 0.84 RECQL (0.67) RECQLHPGDALDH1A1CYP1A2CYP3A4
SCHEMBL24797472 0.81 ALDH1A1 (1.00) HPGDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL1548213 0.77 ALDH1A1 (0.69) HPGDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL30725947 0.77 ALDH1A1 (0.69) HPGDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL4578714 0.75 CLK2 (0.65) RECQLHPGDALDH1A1CYP1A2CYP3A4
SCHEMBL14434248 0.74 ALDH1A1 (1.00) HPGDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL6689373 0.73 ROCK2 (0.58) RECQLHPGDALDH1A1CYP1A2CYP3A4
SCHEMBL23084085 0.73 RECQL (0.66) RECQLHPGDALDH1A1CYP1A2CYP3A4
SCHEMBL7572900 0.73 INSR (0.56) HPGDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL8774349 0.73 ALDH1A1 (0.67) HPGDALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997667-A Pyridinyl compounds of N-carbamoyl-N-thiocarbamoyl- or N-amidino-glycine or beta-alanine useful as sweetening agents UNIVERSITE CLAUDE BERNARD (FR) 1991-03-05 US disclosed
EP-0321369-A1 Heterocyclic sweeteners derived from N-carbamoyl-, N-thiocarbamoyl or N-amidino-glycine or beta-alanine UNIVERSITE CLAUDE BERNARD - LYON 1 (FR) 1989-06-21 EP disclosed