SCHEMBL9879442

SCHEMBL9879442

CSc1nc(=O)c(CCOCc2ccccc2)c(C)[nH]1

nearest known ligand 0.74

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.74
L3MBTL1 Q9Y468 2/20 0.58
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
LMNA P02545 2/20 0.43
POLB P06746 1/20 0.42
HCAR2 Q8TDS4 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
THRB P10828 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 1/20 0.35
STAT1 P42224 1/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9879325 0.85 ALDH1A1 (1.00) ALDH1A1L3MBTL1CYP2C9CYP2C19LMNA
SCHEMBL11079720 0.80 POLB (0.56) ALDH1A1L3MBTL1CYP2C9CYP2C19LMNA
SCHEMBL9879389 0.78 ALDH1A1 (0.52) ALDH1A1L3MBTL1LMNAPOLBTDP1
SCHEMBL9878778 0.71 ALDH1A1 (0.61) ALDH1A1L3MBTL1CYP2C9CYP2C19LMNA
SCHEMBL9879475 0.69 POLB (0.71) ALDH1A1LMNAPOLBMAPTRAB9A
SCHEMBL10735952 0.69 ALDH1A1 (0.73) ALDH1A1L3MBTL1CYP2C9CYP2C19LMNA
SCHEMBL20470604 0.68 ALDH1A1 (0.51) ALDH1A1L3MBTL1CYP2C19HCAR2TDP1
SCHEMBL9829434 0.67 XDH (0.49) ALDH1A1L3MBTL1CYP2C9CYP2C19LMNA
SCHEMBL11458923 0.66 ALDH1A1 (0.52) ALDH1A1L3MBTL1HCAR2RAB9A
SCHEMBL10857015 0.64 LMNA (0.70) ALDH1A1L3MBTL1CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018887-A1 DIAMINOPYRIMIDINE COMPOUNDS SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1991-12-12 WO disclosed