SCHEMBL9900752

SCHEMBL9900752

Cc1onc2cccc(Oc3ccc(N)cc3)c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.41
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
TEAD4 Q15561 1/20 0.40
KDM1A O60341 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
MAPT P10636 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
MITF O75030 1/20 0.39
GAA P10253 1/20 0.39
GFER P55789 1/20 0.39
NLRP1 Q9C000 1/20 0.39
NOD2 Q9HC29 1/20 0.39
TSHR P16473 2/20 0.37
CYP3A4 P08684 1/20 0.37
MAOA P21397 1/20 0.37
APAF1 O14727 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9901077 0.81 ALDH1A1 (0.47) ALDH1A1NCOA1NCOA3TEAD4SMN1; SMN2
SCHEMBL9905767 0.77 KDR (0.43) ALDH1A1NCOA1NCOA3TEAD4SMN1; SMN2
SCHEMBL9905617 0.76 PTGS2 (0.43) ALDH1A1SMN1; SMN2MEN1KMT2APOLB
SCHEMBL15293091 0.73 DCPS (0.48) ALDH1A1NCOA1NCOA3TEAD4KDM1A
SCHEMBL9900459 0.73 AR (0.43) ALDH1A1SMN1; SMN2MEN1KMT2APOLB
SCHEMBL31531346 0.73 KDR (0.56) ALDH1A1NCOA1NCOA3SMN1; SMN2MAPT
SCHEMBL20854306 0.71 TEAD4 (0.56) ALDH1A1NCOA1NCOA3TEAD4SMN1; SMN2
SCHEMBL15284246 0.70 DCPS (0.62) DHFR
SCHEMBL8404508 0.68 ELANE (0.43) TDP1MEN1KMT2AELANEMAPK1
SCHEMBL22830371 0.67 ALDH1A1 (0.50) ALDH1A1NCOA1NCOA3TEAD4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649066-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS Autifony Therapeutics Limited (GB) 2013-10-16 EP disclosed
WO-2012076877-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS AUTIFONY THERAPEUTICS LIMITED (GB) 2012-06-14 WO disclosed