SCHEMBL9904098

SCHEMBL9904098

Cc1nnn(-c2ccccc2F)c1-c1cn(-c2ccc(C(=O)O)cc2)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.36
NOTUM Q6P988 1/20 0.36
TP53 P04637 2/20 0.35
SPR P35270 1/20 0.35
CNR1 P21554 1/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAP4K4 O95819 1/20 0.35
NLRP3 Q96P20 1/20 0.34
GAA P10253 1/20 0.34
GFER P55789 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21402168 0.89 NOTUM (0.38) ALDH1A1HPGDMAPK1NOTUMSPR
SCHEMBL9895440 0.89 IDO1 (0.41) ALDH1A1HPGDHTTBRD4BRD2
SCHEMBL9895332 0.87 SPR (0.38) ALDH1A1NOTUMSPRKDM4AKDM5A
SCHEMBL9895495 0.81 SPR (0.37) SPR
SCHEMBL9896773 0.77 GABRA5 (0.37) HTTSPRGAA
SCHEMBL9895210 0.77 PTGS2 (0.46) PTGS2ALDH1A1HPGDNPC1RAB9A
SCHEMBL21416227 0.75 ALDH1A1 (0.45) ALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL9896578 0.75 LMNA (0.38) PTGS2SPRBRD4BRD2BRD3
SCHEMBL9895387 0.74 CNR2 (0.40) HTTSPRCNR1NPC1RAB9A
SCHEMBL28807048 0.74 PTGS2 (0.39) PTGS2ALDH1A1HPGDHTTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649064-B1 NOVEL TRIAZOLE COMPOUNDS III HOFFMANN LA ROCHE (CH) 2019-10-02 EP claimed
EP-2649064-A1 NOVEL TRIAZOLE COMPOUNDS III F. Hoffmann-La Roche AG (CH) 2013-10-16 EP disclosed
WO-2012076590-A1 NOVEL TRIAZOLE COMPOUNDS III F. HOFFMANN-LA ROCHE AG (CH) 2012-06-14 WO disclosed