SCHEMBL9905376

SCHEMBL9905376

NNC(=O)c1nc2n(c(=O)c1OCc1ccccc1)CC1CCC2(NC(=O)O)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OGFRL1 Q5TC84 1/20 0.35
FAAH O00519 4/20 0.35
CNR2 P34972 4/20 0.35
MAPT P10636 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HDAC6 Q9UBN7 1/20 0.33
CNR1 P21554 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
NPC1 O15118 1/20 0.32
HPGD P15428 1/20 0.32
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
S1PR5 Q9H228 1/20 0.31
SGMS2 Q8NHU3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14214193 0.92 TSHR (0.36) OPRM1OPRD1OPRK1OGFRL1FAAH
SCHEMBL9905325 0.85 SIGMAR1 (0.35) CNR2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL9921626 0.84 TLR2 (0.36) OPRD1OPRK1MAPTALDH1A1
SCHEMBL9905089 0.84 CHRM4 (0.34) CNR2MAPTALDH1A1CNR1KMT2A
SCHEMBL9905103 0.84 RORC (0.36) FAAHCNR2ALDH1A1GAA
SCHEMBL14122239 0.83 MAPT (0.33) OPRM1OPRD1OPRK1OGFRL1FAAH
SCHEMBL9905086 0.82 HPGD (0.39) MAPTHPGDKDM4ESMN1; SMN2
SCHEMBL9905381 0.82 CTSL (0.39) ALDH1A1HPGDSMN1; SMN2
SCHEMBL14214197 0.79 ALDH1A1 (0.34) CNR2MAPTALDH1A1KMT2AMEN1
SCHEMBL14214192 0.78 ALDH1A1 (0.34) CNR2MAPTALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649074-A1 HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2013-10-16 EP disclosed
WO-2012078844-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed