SCHEMBL9905381

SCHEMBL9905381

N#CC(Cc1ccc(F)cc1)NC(=O)c1nc2n(c(=O)c1OCc1ccccc1)CC1CCC2(NC(=O)O)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.39
GPR34 Q9UPC5 2/20 0.34
YAP1 P46937 1/20 0.34
CTSC P53634 7/20 0.33
CTSS P25774 1/20 0.33
CHRM4 P08173 1/20 0.33
CTSK P43235 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
DPP4 P27487 1/20 0.32
FAP Q12884 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
DPP9 Q86TI2 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16130153 0.94 CTSL (0.38) CTSLGPR34YAP1CTSCCTSS
SCHEMBL16130199 0.88 CTSL (0.36) CTSLYAP1CTSSCTSK
SCHEMBL14122652 0.87 CTSL (0.36) CTSLGPR34YAP1CTSCCTSS
SCHEMBL9905325 0.84 SIGMAR1 (0.35) CTSLCHRM4ALDH1A1HPGDSMN1; SMN2
SCHEMBL9905089 0.83 CHRM4 (0.34) CTSLCHRM4ALDH1A1HPGDSMN1; SMN2
SCHEMBL9905376 0.82 OPRM1 (0.35) ALDH1A1HPGDSMN1; SMN2
SCHEMBL1669098 0.79 CTSL (0.37) CTSLGPR34YAP1CTSCCTSS
SCHEMBL14214197 0.78 ALDH1A1 (0.34) CTSLYAP1CHRM4ALDH1A1HPGD
SCHEMBL14214192 0.77 ALDH1A1 (0.34) CTSLCTSSCHRM4ALDH1A1HPGD
SCHEMBL9905364 0.76 MAPT (0.35) ALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649074-A1 HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2013-10-16 EP disclosed
WO-2012078844-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed