SCHEMBL990705

SCHEMBL990705

CN(C)CCOC(=O)[C@@H](N)CCC(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 2/20 0.46
PMP22 Q01453 2/20 0.46
ALOX15 P16050 1/20 0.46
KMT2A Q03164 1/20 0.46
CHRM1 P11229 3/20 0.44
CHRNB2 P17787 2/20 0.44
CHRNA4 P43681 2/20 0.44
CHRM2 P08172 2/20 0.44
CHRM3 P20309 2/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
DNM1 Q05193 1/20 0.40
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
PHLPP2 Q6ZVD8 1/20 0.38
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4560462 0.98 BLM (0.44) BLMPMP22ALOX15KMT2ACHRM1
SCHEMBL3032152 0.86 DNM1 (0.51) BLMPMP22CHRM1CHRNB2CHRNA4
SCHEMBL24160467 0.82 CHRM1 (0.47) CHRM1CHRNB2CHRNA4CHRM2CHRM3
SCHEMBL8009500 0.81 ALOX15 (0.56) BLMPMP22ALOX15KMT2ACHRNB2
SCHEMBL2305262 0.80 ALOX15 (0.50) BLMPMP22ALOX15KMT2ADPP4
SCHEMBL28643800 0.80 KMT2A (0.50) BLMPMP22ALOX15KMT2ADPP4
SCHEMBL15198720 0.80 DNM1 (0.39) BLMPMP22CHRM1CHRNB2CHRNA4
SCHEMBL398286 0.78 ALOX15 (0.52) BLMPMP22ALOX15KMT2ADPP4
SCHEMBL8581073 0.77 NOD1 (0.49) BLMPMP22ALOX15KMT2ADPP4
SCHEMBL8749113 0.77 NOD1 (0.49) BLMPMP22ALOX15KMT2ADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101808599-B Possesses the foley's tube launching guard member INVATEC TECHNOLOGY CENTER GMBH (CH) 2016-01-27 CN disclosed
WO-2014176458-A2 BIORESORBABLE BIOPOLYMER ANASTOMOSIS DEVICES TRUSTEES OF TUFTS COLLEGE (US) 2014-10-30 WO disclosed
CN-103930158-A Balloon assembly with controllably variable topography GORE & ASS 2014-07-16 CN disclosed
CN-101808676-B Improved drug-coated pharmaceutical products, their manufacture and use INVATEC TECHNOLOGY CT GMBH 2014-06-04 CN disclosed
CN-103665170-A Peptide therapeutic conjugates and uses thereof ANGIOCHEM INC 2014-03-26 CN disclosed
EP-2456573-A1 MEDICAL DEVICE COATING SYSTEM Boston Scientific Scimed, Inc. (US) 2012-05-30 EP disclosed
WO-2011011433-A1 MEDICAL DEVICE COATING SYSTEM BOSTON SCIENTIFIC SCIMED, INC. (US) 2011-01-27 WO disclosed
EP-2086600-A2 STENTS WITH DRUG ELUTING COATINGS Boston Scientific Limited (BB) 2009-08-12 EP disclosed
EP-2051750-A2 COATINGS FOR MEDICAL DEVICES COMPRISING A THERAPEUTIC AGENT AND A METALLIC MATERIAL Boston Scientific Limited (Barbados Home Office) (BB) 2009-04-29 EP disclosed
WO-2007130422-A9 NON-STICKY COATINGS WITH THERAPEUTIC AGENTS FOR MEDICAL DEVICES BOSTON SCIENT LTD (BB) 2009-02-05 WO disclosed
EP-2019697-A2 NON-STICKY COATINGS WITH THERAPEUTIC AGENTS FOR MEDICAL DEVICES Boston Scientific Limited (BB) 2009-02-04 EP disclosed
EP-1979013-A2 COATED MEDICAL DEVICES AND METHODS OF MAKING THE SAME Boston Scientific Limited (BB) 2008-10-15 EP disclosed
WO-2008066656-A2 STENTS WITH DRUG ELUTING COATINGS BOSTON SCIENTIFIC LIMITED (BB) 2008-06-05 WO disclosed
WO-2008002586-A2 COATINGS FOR MEDICAL DEVICES COMPRISING A THERAPEUTIC AGENT AND A METALLIC MATERIAL BOSTON SCIENTIFIC LIMITED (BB) 2008-01-03 WO disclosed
WO-2007130422-A2 NON-STICKY COATINGS WITH THERAPEUTIC AGENTS FOR MEDICAL DEVICES BOSTON SCIENTIFIC LIMITED (BB) 2007-11-15 WO disclosed
EP-1811922-A1 SYSTEM AND METHOD FOR DELIVERING A BIOLOGICALLY ACTIVE MATERIAL TO A BODY LUMEN Boston Scientific Limited (BB) 2007-08-01 EP disclosed
WO-2007084361-A2 COATED MEDICAL DEVICES AND METHODS OF MAKING THE SAME BOSTON SCIENTIFIC LIMITED (BB) 2007-07-26 WO disclosed
WO-2006044038-A1 SYSTEM AND METHOD FOR DELIVERING A BIOLOGICALLY ACTIVE MATERIAL TO A BODY LUMEN BOSTON SCIENTIFIC LIMITED (BB) 2006-04-27 WO disclosed
EP-1392756-A2 LIPID-POLYMER-CONJUGATES Yamanouchi Europe B.V. (NL) 2004-03-03 EP disclosed
WO-2002098951-A2 LIPID-POLYMER-CONJUGATES YAMANOUCHI EUROPE B.V. (NL) 2002-12-12 WO disclosed